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2-[4-(4-methylpyrimidine-5-carbonyl)piperazin-1-yl]-1-(pyrrolidin-1-yl)ethan-1-one
N-benzyl-2-(pyridin-3-yl)piperidine-1-sulfonamide
1-benzyl-N-ethyl-5-[(2-hydroxyethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[(4-fluorophenyl)methyl]-5-[5-(methoxymethyl)furan-2-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
4-(3-methylbut-2-en-1-yl)-3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]piperazin-2-one
5-(2,4-dimethoxyphenyl)-N-[(3,5-dimethoxyphenyl)methyl]-1,2,4-triazin-3-amine
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyrazine
N-[(3S)-1-benzylpyrrolidin-3-yl]-4-methyl-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
N-[2-(2,4-dimethoxyphenyl)ethyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2,6-dimethyl-4-(3-phenoxyazetidine-1-carbonyl)quinoline
7-[(2,3-dimethyl-1H-indol-7-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-methyl-2-{4-[2-(propan-2-yloxy)phenyl]-1H-pyrazol-1-yl}acetamide
2-{3-cyclopropyl-5-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-1,2,4-triazol-1-yl}pyridine
(1S,3R)-N-cyclohexyl-3-[3-(6-oxo-1,4,5,6-tetrahydropyridazin-3-yl)propanamido]cyclopentane-1-carboxamide
2-(4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl)ethan-1-ol
1-cyclohexyl-4-(3,3,3-trifluoro-2-hydroxypropanoyl)piperazin-2-one
1-{3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(morpholin-4-yl)phenyl}ethan-1-one
1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-4-(furan-2-carbonyl)-1,4-diazepane
1-ethyl-2-{[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
5-[1-(5-methyl-2-phenylfuran-3-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-chloro-4-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}benzamide
3-cyclopentaneamido-N-(1-methanesulfonylpiperidin-4-yl)benzamide
1-methyl-4-{2-[3-(2-methylpropyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]ethyl}piperidine
3-[1-({5-ethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperidin-4-yl]-1,3-oxazolidin-2-one
3-{2-[3-(oxolan-2-ylmethyl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-indole
1-(1-methylcyclopropanecarbonyl)-4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine
1-(4-cyano-2-fluorophenyl)-3-(2-methoxyethyl)-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
2-[3-methyl-4-({methyl[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)-1H-pyrazol-1-yl]ethan-1-ol
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl]-3,5-dimethoxybenzamide
(3S)-1-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-ol
2-cyclopentyl-9-(2-phenoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
3-{[5-(cyclohex-3-en-1-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine
N,1,3-trimethyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-[3-(1H-1,3-benzodiazol-2-yl)propanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-[4-(2-methylpropyl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}oxan-4-amine
N-[(3S,7S,8aS)-3-(cyclohexylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,5-difluorobenzamide
methyl 1-(benzyloxy)-8-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
5-(4-chloro-2,6-dimethoxyphenyl)-1-methyl-1H-1,2,3,4-tetrazole
1-(furan-2-ylmethyl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)piperidine-3-carboxamide
3-chloro-6-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}pyridazine
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(oxan-4-ylmethyl)acetamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[2-(2-methoxyphenyl)ethyl]amine
7-[cyclohexyl(methoxy)methyl]-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1H-imidazol-2-yl}-6,8-dimethyl-1,2-dihydroquinolin-2-one
1-{3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl}piperidine-3-carbonitrile
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-{[5-(hydroxymethyl)furan-2-yl]methyl}pyrrolidin-3-yl]methanol