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3-[5-(3-methoxy-5-methylthiophene-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
1-{4-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
2-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
2-methoxy-6-[2-(trifluoromethyl)morpholine-4-carbonyl]phenol
6-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
N,N,4-trimethyl-5-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine-1-carbonyl)pyrimidin-2-amine
1-{4-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]phenyl}piperidine
4,4,4-trifluoro-N-[(3R,4S)-4-(3-methoxyphenyl)-1-methylpyrrolidin-3-yl]butanamide
7-(1,3-benzothiazol-2-yl)-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S,4S)-4-[3-(dimethyl-1,2-oxazol-4-yl)propanamido]-N-ethyl-1-(2-methoxyethyl)pyrrolidine-2-carboxamide
1-[1-(3-phenylphenyl)piperidin-4-yl]piperidin-4-amine
1-(2-methyl-7-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl)pyrrolidine
3-[({1-[(2,3-difluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)(methyl)amino]propanamide
(1-{[1-(4-ethyl-5-methylthiophene-3-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
2,4-dimethyl-N-[2-(piperidin-1-yl)ethyl]-1,3-oxazole-5-carboxamide
5-[(3-cyclohexylpyrrolidin-1-yl)methyl]-3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazole
N-(2-hydroxyethyl)-3,5,7-trimethyl-N-(1,3-thiazol-2-ylmethyl)-1H-indole-2-carboxamide
3-amino-N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)-1H-1,2,4-triazole-5-carboxamide
5-[(4-fluorophenyl)methyl]-3-[2-(1H-imidazol-1-yl)ethyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
2,5-dimethoxy-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
N-({3-[4-fluoro-3-(hydroxymethyl)phenyl]phenyl}methyl)propanamide
2-(4-benzoylpiperazine-1-carbonyl)-N-propylaniline
9-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[(pyridin-3-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-methyl-3-propyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-pyrazole-5-carboxamide
4-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-methyl-2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}quinoline
1-[2-(cyclopent-2-en-1-yl)acetyl]-4-(3-methylphenoxy)piperidine-4-carboxylic acid
methyl 4-(4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)benzoate
methyl 4-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
1,3,5-trimethyl-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}-1H-pyrazole-4-sulfonamide
1-[(2-fluorophenyl)methyl]-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-6-oxopiperidine-3-carboxamide
6-[1-(1H-indol-1-yl)propan-2-yl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-[(2,4-difluorophenyl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
1-[(3-{1,6-dimethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1,2-oxazol-5-yl)methyl]piperidin-4-ol
ethyl 3-[(4-fluorophenyl)methyl]-1-[4-(2-oxopiperidin-1-yl)butanoyl]piperidine-3-carboxylate
1-(3-chlorophenyl)-4-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazine
2-[2-(3-fluorophenoxymethyl)pyrimidin-4-yl]pyridine-4-carboxylic acid
5-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-2-(propan-2-yl)-1,3-benzoxazole
2-{4-[4-(3,3-dimethylpyrrolidine-1-carbonyl)-7,8-dimethylquinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
1,9-dimethyl-4-{[2-(propylsulfanyl)pyrimidin-5-yl]methyl}-1,4,9-triazaspiro[5.5]undecane
(3aR,6aR)-2-(2-hydroxyethyl)-5-(1,3-thiazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(4-ethylpiperazin-1-yl)methyl]-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
1-(2-aminoethyl)-N-(5-methyl-2-pentanamidophenyl)-1H-1,2,3-triazole-4-carboxamide
1-benzyl-8-(propan-2-yl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-oxo-1-(pyridin-2-ylmethyl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)pyrrolidine-3-carboxamide
5-methyl-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-1-propyl-1H-pyrazole-4-carboxamide
2-[5-(1-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
N-(3-methoxyphenyl)-3-[1-(3-phenylpropyl)piperidin-4-yl]propanamide