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N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
1-[(2-fluoro-5-methylphenyl)methyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
[({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)sulfamoyl]dimethylamine
3-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-ol
1-[1-(4-methoxy-3-methylbenzoyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
6-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]propanamide
N-(3-{[(2-chlorophenyl)methyl]sulfanyl}propyl)-5-methyl-1,3,4-oxadiazol-2-amine
3-fluoro-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
1-(2-chloroprop-2-en-1-yl)-3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-6,7-dimethoxy-1,2-dihydroquinolin-2-one
N,2,3-trimethyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
(2R,3S,6R)-5-(2-fluorobenzoyl)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(1R,5R)-6-benzyl-3-(5-ethyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{3-oxa-9-azaspiro[5.5]undecan-9-yl}-2-oxo-N-propylacetamide
3-[(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-1,2,3-triazol-1-yl)methyl]piperidine
N-benzyl-N-methyl-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
4-hydroxy-N-(2-methoxyethyl)-2-phenyl-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
7-(5-chloropyridin-2-yl)-4-(furan-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S)-2-[(4-cyclopentylpyrimidin-2-yl)amino]-3-methylbutanamide
methyl[(3-methyl-1,2-oxazol-5-yl)methyl](4,5,6,7-tetrahydro-2H-indazol-3-ylmethyl)amine
2-[4-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(2-methylpropyl)piperazin-2-yl]ethan-1-ol
2-[3-(2-methylpropyl)-5-[pyridin-3-yl(pyrrolidin-1-yl)methyl]-1H-1,2,4-triazol-1-yl]pyridine
3-(1-methyl-1H-pyrrol-2-yl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-pyrazole-5-carboxamide
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-[1-(1,3-thiazol-5-yl)ethyl]propanamide
(2R)-1-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}pyrrolidine-2-carboxamide
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-[2-(5-methyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
2-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-1,2,3,4-tetrahydroisoquinoline
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(2-fluorophenyl)propanamide
7-(cyclopropylmethyl)-N-(2-methoxy-5-methylphenyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
2-oxo-6-(propan-2-yl)-N-[2-(4-sulfamoylphenyl)ethyl]-1,2-dihydropyridine-3-carboxamide
1-ethyl-3-(naphthalen-1-ylmethyl)-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[3-(4-methyl-1,3-thiazol-5-yl)propyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
4-{1-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1H-imidazol-2-yl}-2,1,3-benzoxadiazole
2-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-1,3-thiazole-4-carboxamide
3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-N-(2-ethylphenyl)piperidine-1-carboxamide
4-hydroxy-2-methyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]pyrimidine-5-carboxamide
[4-(3,4,7-trimethyl-1H-indole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
1-[(3-methylphenyl)methyl]-4-[1-(1-methylpiperidin-4-yl)pyrrolidine-2-carbonyl]piperazine
3-cyclopropyl-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-1-[3-(azepane-1-carbonyl)phenyl]urea
4-{1-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]piperidin-3-yl}benzoic acid
2-(2,2-dimethylpropanamido)-N,5-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]thiophene-3-carboxamide
15-methyl-13-oxo-N-(prop-2-en-1-yl)-9-(thiophen-3-yl)-4-(trifluoromethyl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}urea
4-(2,4-dioxoimidazolidin-1-yl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}benzamide
1-{1-[6-(piperidin-4-yl)pyrimidin-4-yl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-hydroxy-5-methyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)benzamide
N-methyl-4-{[(4-methylphenyl)methyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
1-{1-[6-(dimethylamino)pyrazin-2-yl]piperidin-4-yl}piperidin-4-ol