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3-methoxy-2-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
5-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
5-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-(piperazin-1-yl)propan-1-one
(4aS,8aR)-1-(2-methylpropyl)-6-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
(2S)-1-{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidine-2-carboxamide
9-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1,4,9-triazaspiro[5.5]undecan-5-one
2-[1-(4,6-dimethylpyridine-3-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
(3S,4R)-1-[2-(benzenesulfonyl)ethyl]-4-methylpiperidine-3,4-diol
(3aS,6aR)-5-(5-ethyl-1,3-oxazole-4-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-[2-(1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]morpholine
7-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
5-(furan-2-yl)-3-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]methyl}-1,2-oxazole
5-[(2,2-dimethylpyrrolidin-1-yl)methyl]-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-{1-[(2-fluorophenyl)methyl]-4-[(8-methoxy-2H-chromen-3-yl)methyl]piperazin-2-yl}ethan-1-ol
(3S,7S)-5-[5-(methoxymethyl)furan-2-carbonyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-[2-(2-ethylphenoxy)ethyl]-N-methyl-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2-[4-(3-chloropyridin-2-yl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
1-[1-(1-tert-butyl-3-methyl-1H-1,2,4-triazol-5-yl)ethyl]pyrrolidin-2-one
3-(3-hydroxy-1,2-oxazol-5-yl)-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
2-amino-6-(2,4-dimethylphenyl)-4-[5-(hydroxymethyl)furan-2-yl]pyridine-3-carbonitrile
7-{2-[4-(3-methylphenyl)piperazin-1-yl]acetyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-(3-fluorophenoxymethyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
(2R)-2-methoxy-2-phenyl-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
methyl 2-{3-oxo-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
1-[(2-chlorophenyl)methyl]-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-ethyl-4-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
2-(2-chlorophenyl)-N-[2-(dimethylamino)ethyl]-N-ethyl-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-[(cyclopropylmethyl)sulfanyl]ethan-1-one
methyl({[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}){[3-(trifluoromethyl)phenyl]methyl}amine
3-{2-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-4-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
3-methyl-7-[3-(2-methylphenoxy)azetidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
2-{[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}-4-fluorophenol
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[3-(propan-2-yloxy)propyl]-1H-1,3-benzodiazole-5-carboxamide
2-(2,3-dihydro-1H-isoindol-2-yl)-1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)ethan-1-one
2-(2-methylpropyl)-8-(pyrimidin-5-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-(2-methyl-1-{2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-1-oxopropan-2-yl)acetamide
(1S,4S)-2-(2-chlorophenyl)-5-(furan-3-ylmethyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
2-cyclopropyl-5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
2-[2-(1H-imidazol-4-yl)ethyl]-8-[(3E)-pent-3-enoyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(5-carbamoyl-2-methylphenyl)-2-[2-(4-methylpiperazin-1-yl)ethyl]piperidine-1-carboxamide
2-methyl-6-{[1-(2-methylphenyl)piperidin-4-yl]amino}heptan-2-ol
{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(3S,4R)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)sulfonyl]-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
N-({1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}methyl)thiophene-2-sulfonamide
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(2,3,4,9-tetrahydro-1H-carbazole-8-carbonyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-(trimethyl-1H-pyrazol-1-yl)acetamide