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2-methoxy-1-{4-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]-1,4-diazepan-1-yl}ethan-1-one
2-benzyl-8-[2-(1H-imidazol-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-{[(2S,4S)-4-fluoro-1-[3-(2-oxoazepan-1-yl)propanoyl]pyrrolidin-2-yl]methyl}-3-(methylsulfanyl)propanamide
[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl){[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
[4-(3-phenylpropyl)-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]methanol
4-(3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}propanoyl)-3-ethyl-3-methylpiperazin-2-one
8-[3-(3-ethylphenoxy)azetidine-1-carbonyl]quinoline
6-fluoro-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-[(2-fluoro-5-methoxyphenyl)methyl]-9-oxa-2-azaspiro[5.5]undecane
4-(3-hydroxy-3-methylbutyl)-N-[1-(6-methylpyridin-2-yl)ethyl]benzamide
4-(2-methyl-1H-imidazol-1-yl)-1-[3-(thiophen-2-yl)propanoyl]piperidine-4-carboxylic acid
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(pyridin-3-yl)acetyl]pyrrolidine-3-carboxylic acid
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-(2,3-dihydro-1H-inden-2-yl)acetamide
3-hydroxy-1-(2-methoxyethyl)-3-({[(3-methyl-1-benzofuran-2-yl)methyl]amino}methyl)piperidin-2-one
N-{[5-(3-chlorophenyl)furan-2-yl]methyl}-2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[2-(pyridin-3-yloxy)propyl]amine
propyl 4-{3-[(pyridin-3-ylmethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxylate
2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propan-1-ol
2-[5-(ethylsulfanyl)thiophene-2-carbonyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
4-phenyl-2-[1-(prop-2-en-1-yl)-1H-imidazol-2-yl]-1,3-thiazole
methyl 2-[4-(4-phenyl-5-propyl-1H-imidazol-1-yl)piperidin-1-yl]acetate
4-(1-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}azetidin-3-yl)pyridine
(3R,4R)-4-(hydroxymethyl)-1-(2-phenylquinoline-4-carbonyl)piperidin-3-ol
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethylbenzamide
3-{[2-(morpholin-4-ylmethyl)-1,4-oxazepan-4-yl]methyl}benzoic acid
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]pyrrolidine-1-carboxamide
N-[(3R,4S)-1-(2-ethoxyethyl)-4-phenylpyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
(1S,5R)-6-[(6-methylpyridin-2-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
methyl N-[2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]carbamate
2-[(2-{ethyl[3-(morpholin-4-yl)propyl]carbamoyl}phenyl)amino]acetic acid
N-methyl-5-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyrimidin-2-amine
N-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-4-(pyridin-4-yl)piperazine-1-carboxamide
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
[(3-methyl-1H-pyrazol-5-yl)methyl](propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amine
1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-[2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]azetidin-3-ol
2-({[1-(hydroxymethyl)cyclopropyl]methyl}(methyl)sulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-{[methyl(2-phenylethyl)amino]methyl}pyridine-3-carboxylic acid
3-(1-ethyl-1H-imidazol-2-yl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
5-(1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
N-ethyl-5-[(4-hydroxypiperidin-1-yl)methyl]-N-(1-phenylethyl)-1,2-oxazole-3-carboxamide
1-[(2-methoxyphenyl)methyl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
1-[1-(2,3-dihydroxypropyl)piperidin-4-yl]butan-1-one
2-amino-7-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-ethyl-3-(propan-2-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1H-pyrazole-5-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
4-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-methylquinoline
(2S,4S)-4-amino-1-{4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butanoyl}pyrrolidine-2-carboxylic acid