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3-(3-chloro-1,2-oxazol-5-yl)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
2-(3-methoxypropyl)-9-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
8-[(2-butyl-1H-imidazol-4-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(2-{2-[1-(3-methoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
5-[(5-fluoro-2-methoxyphenyl)methyl]-2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
methyl 2-{4-[2-(1H-1,3-benzodiazol-1-yl)propanoyl]-3-methyl-2-oxopiperazin-1-yl}acetate
1-methyl-3-phenyl-8-[2-(pyridin-4-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
(3-{2-[1-(3-ethoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
dimethyl({4-[2-methyl-5-(propan-2-yl)pyrimidin-4-yl]phenyl}methyl)amine
2-{3-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidine-1-carbonyl]phenoxy}acetamide
4-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethyl-4-oxobutanamide
8-(2-propyl-1,3-thiazole-4-carbonyl)-1-oxa-8-azaspiro[4.5]decane
1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}azepane
6-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
4-[3-(4-fluorophenyl)-1H-pyrazole-5-amido]oxane-4-carboxylic acid
{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(pyrazin-2-yl)ethyl]amine
(1R,4S)-2-(2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carbonyl)-2-azabicyclo[2.2.1]heptane
3-[methyl({3-[3-(3-methylphenoxy)azetidin-1-yl]-3-oxopropyl})amino]-1λ6-thiolane-1,1-dione
3-methyl-N-{2-methyl-5-[2-(methylamino)acetamido]phenyl}benzamide
(3S,4S)-4-cyclopropyl-1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]pyrrolidine-3-carboxylic acid
2-{2-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
3-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}-1H-pyrazol-5-amine
2-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}-6-methoxyphenol
1-[3-(1H-imidazol-2-yl)benzoyl]-3-[2-(2-methylphenyl)ethyl]piperidine
(1S,5R)-3-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{1-[(3-hydroxyphenyl)methyl]piperidin-4-yl}oxolane-3-carboxamide
N3-butyl-N5-[(5-fluoro-2-methylphenyl)methyl]-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
8-(2-hydroxyacetyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-{3-[4-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}pyrrolidin-3-yl)pyridin-2-yl]phenyl}ethan-1-one
1-{2-[({3-[2-hydroxy-3-(morpholin-4-yl)propoxy]phenyl}methyl)amino]ethyl}pyrrolidin-2-one
3-(4-chloro-1H-pyrazol-1-yl)-N-methyl-N-(quinolin-5-ylmethyl)propanamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
4-[(2-ethylpyrimidin-5-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-4-methylpentane-1,2-dione
2,5-dimethyl-N-{3-[methyl(phenyl)amino]propyl}-1,3-thiazole-4-carboxamide
2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-6-methylpyridine-4-carboxylic acid
2-(phenylamino)-N-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]pyrimidine-5-carboxamide
3-methoxy-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1,2-dihydropyridin-2-one
7-(cyclobutylmethyl)-2-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N,N-dimethyl-3-({3-[(oxolan-3-yl)sulfamoyl]phenyl}formamido)propanamide
4,6-dimethyl-2-oxo-N-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-1,2-dihydropyridine-3-carboxamide
N-[(1-{2-[(3-chlorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperidin-3-yl)methyl]acetamide
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-(propan-2-yl)pyrimidine
1-[2-(3-fluorophenyl)ethyl]-5-[4-(2-methoxyethyl)piperazine-1-carbonyl]piperidin-2-one
2,4-dimethyl-N-{4-[(2-methylprop-2-en-1-yl)oxy]phenyl}-3-oxopiperazine-1-carboxamide
2-[(isoquinolin-5-yloxy)methyl]-N-methyl-N-(oxolan-2-ylmethyl)-1,3-oxazole-4-carboxamide
1-{2-[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]ethyl}-4-(propan-2-yl)piperazine
1-[1'-(1-methyl-1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
3-[(2-hydroxyethyl)(methyl)sulfamoyl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]benzamide
1-{4-[2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}-2,2-diphenylethan-1-one