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N-{4-[1-(5-oxo-1-propylpyrrolidin-3-yl)-4-phenyl-1H-imidazol-5-yl]phenyl}acetamide
5-methoxy-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}furan-2-carboxamide
1-[3-(azepan-1-yl)-2-hydroxypropyl]-3-(1H-indazol-6-yl)urea
N-{1-[1-(2-hydroxy-4-methylpentanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-[2-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-1-phenylcyclopropane-1-carboxamide
3-methyl-1-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperidine
6-(2,5-dimethoxyphenyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
(3R,4S)-1-(2-methanesulfonylethyl)-4-phenylpyrrolidin-3-amine
N2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N4,6-dimethylpyrimidine-2,4-diamine
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(prop-2-en-1-yl)acetamide
5-{[(5-methylpyrazin-2-yl)methyl]carbamoyl}thiophene-2-carboxylic acid
(1S,5R)-6-(cyclobutylmethyl)-3-[(3-methylquinoxalin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2,5-dimethyl-N-[1-(thiophen-3-yl)propan-2-yl]-1,3-thiazole-4-carboxamide
4-(4-phenyl-1-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-imidazol-5-yl)phenol
N-(1-benzylpyrrolidin-3-yl)-5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-(2-hydroxy-3-methoxypropyl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-2-(propan-2-yl)pyrimidine-4-carboxamide
3-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1,4-diazepane
1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-ol
2-methoxy-4-({[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenol
(2S,4S)-4-amino-N,N-diethyl-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}pyrrolidine-2-carboxamide
5,8-dimethyl-2-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}quinolin-4-ol
(4aS,7aR)-1-(5-hydroxypyrazine-2-carbonyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,4-dichloro-3-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}phenol
1-acetyl-N-[(5-tert-butyl-1,3-benzoxazol-2-yl)methyl]piperidine-4-carboxamide
2-methyl-4-(3-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}phenyl)butan-2-ol
3-[(2R,3R,6R)-5-(6-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2,5-dimethylphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[4-(2-cyclopropyl-1H-imidazol-1-yl)phenyl]-1H-1,2,3,4-tetrazole
1-benzyl-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methylpiperidin-4-amine
9-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-6-oxa-9-azaspiro[4.5]decane
2-cyclopropyl-8-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(4-{4-[(2,3-dihydro-1H-inden-2-yl)amino]piperidin-1-yl}benzoyl)piperidin-3-ol
N-ethyl-N-(oxolan-2-ylmethyl)-1-(pyrazine-2-carbonyl)piperidin-4-amine
2,4-dimethyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)pyrimidine-5-carboxamide
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
N-[(3R,4R)-1-[3-(4-fluorophenoxy)propyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
(3R,5S)-5-{4-[4-(benzyloxy)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
1-[3-(2,5-difluorobenzoyl)piperidin-1-yl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propan-1-one
1-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-4-(1H-pyrazol-3-yl)piperidine
3-[(3R,4S)-1-(1-methyl-1H-indole-3-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
7-(1-benzothiophen-3-yl)-4-cyclobutanecarbonyl-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1S,5R)-3-(oxan-4-yl)-6-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1,7-dimethyl-2,4-dioxo-1H,2H,3H,4H-pyrido[2,3-d]pyrimidine-5-carboxamide
1-(4-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methoxy}phenyl)propan-1-one
N,N-dimethyl-3-{2-methyl-1H-imidazo[4,5-b]pyridin-6-yl}aniline
(3S,4S)-4-cyclopropyl-1-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]pyrrolidine-3-carboxylic acid
N-({8-[3-(4-fluorophenyl)benzoyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)pyridine-2-carboxamide