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1-cyclopentyl-3-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
4-methyl-2-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]-1H-1,3-benzodiazole
2-{[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]amino}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[2,4-dioxo-1-(2-phenylethyl)-8-{[2-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
3-[4-(3-chlorophenyl)piperazin-1-yl]-5-(3-fluorophenyl)-1,2,4-triazine
N-{[7-(cyclopent-1-ene-1-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1H-indole-2-carboxamide
2-({[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amino}methyl)phenol
phenyl (7S,9aR)-7-[(1R)-1-hydroxyethyl]-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
(3R,4R)-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-cyclobutanecarbonylpyrrolidine-2-carboxamide
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-(pyridine-2-carbonyl)-1,4-diazepane
7-(5-methylthiophen-2-yl)-4-(pyrimidin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl[(3-{2-[4-(1-methylpiperidine-2-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](thiophen-2-ylmethyl)amine
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
N-(1,2-oxazol-3-ylmethyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
3-(4-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)phenol
8-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
2-(3-fluoropyridin-4-yl)-N-(propan-2-yl)pyridine-4-carboxamide
1-(2-methoxyphenyl)-4-(2-methoxypyridine-4-carbonyl)-5-methylpiperazin-2-one
N-[1-(pyrazin-2-yl)piperidin-4-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
4-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)azetidin-3-yl]morpholine
2-(3-fluorophenyl)-5-(thiomorpholine-4-carbonyl)-1,3-benzoxazole
1-cyclohexyl-3-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)-1-(pyridin-4-ylmethyl)urea
1-({2-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)piperidin-4-ol
8-benzoyl-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
(3S,4S)-1-[(6-methoxy-2H-chromen-3-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
5-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-N-methylpyrimidin-2-amine
1-{1'-[(5-acetylthiophen-3-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
5-{1-[(2-hydroxy-5-methylphenyl)methyl]piperidin-4-yl}-5-(pyridin-3-yl)imidazolidine-2,4-dione
5-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}pyrimidin-2-amine
N-(3-chlorophenyl)-2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N,4,6-trimethyl-2-oxo-N-(quinoxalin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]-2,3,4,9-tetrahydro-1H-carbazole-6-carboxamide
{1-[(3-methyl-1H-pyrazol-5-yl)methyl]-3-propylpiperidin-3-yl}methanol
1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-3-(methoxymethyl)piperidine
(1S,5R)-6-(3-ethoxybenzoyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-{2-[1-cyclohexyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
(4aS,8aS)-2-{2-[(4-methylphenyl)methyl]benzoyl}-decahydro-2,7-naphthyridin-4a-ol
[3-ethyl-1-(2-phenoxyethyl)piperidin-3-yl]methanol
4-(3,4-dimethylphenyl)-3-(1H-pyrazol-5-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[4-(1-ethyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]-N-[(4-methylphenyl)methyl]propanamide
{1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1-methyl-6-oxo-N-(pyridin-4-ylmethyl)-1,6-dihydropyridazine-3-carboxamide
1-[(4-methylphenyl)methyl]-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-2-one
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-4-propylpyrimidine
3-{[4-ethyl-5-oxo-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}-N,N-dimethyl-1,2,4-oxadiazole-5-carboxamide
1-(2-{4-[(2-methyl-1H-imidazol-4-yl)methyl]morpholin-2-yl}ethyl)-3-(propan-2-yl)urea