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1-(2,3-dihydro-1H-indene-5-carbonyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-(4-{[4-(2-aminoethyl)phenyl]methyl}-1,4-diazepan-1-yl)-2,2,2-trifluoroethan-1-one
N-{4-[4-(hydroxymethyl)phenyl]-2-methoxyphenyl}acetamide
N-cyclopropyl-1-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)piperidine-4-carboxamide
5-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1-(prop-2-en-1-yl)piperidin-2-one
3-hydroxy-3-({[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N-(2-methyl-1-{7-[(2,4,5-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)methanesulfonamide
N,1-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H-indole-4-carboxamide
1-methyl-5-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-3-(propan-2-yl)-1H-pyrazole
{5-[1-(1-benzylpyrrolidin-3-yl)-1H-1,2,3-triazol-4-yl]furan-2-yl}methanol
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methylacetamide
3-methyl-N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(1,4-dioxan-2-ylmethyl)-N-methylacetamide
1-(2-methoxyacetyl)-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)piperidine-3-carboxamide
N-[(2R,3R)-2-methoxy-1'-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,3,5-trimethyl-1H-indole-2-carboxamide
N-[(4-hydroxyphenyl)methyl]-1-methyl-3-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
3-(4-methoxyphenyl)-3-phenyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}propanamide
methyl({[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]propanamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
8-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
4-{3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]propoxy}benzamide
3-(3,4-dimethoxybenzoyl)-1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperidine
(3S,4R)-4-(4-fluorophenyl)-1-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-3-carboxylic acid
N-(adamantan-1-yl)-3-{[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
2-[5-(4-methyl-1,3-oxazol-5-yl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl]acetic acid
N-[2-(3-methoxyphenyl)phenyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-2,6-dimethylquinoline
N-[(1S,2R)-2-aminocyclobutyl]-2-[(1-ethyl-1H-indol-3-yl)sulfanyl]acetamide
5-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1H-imidazol-2-yl}-6-methylquinoline
(3S,9aR)-3-benzyl-8-(2-methoxybenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[3-(1H-indol-1-yl)propyl]-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
3-ethyl-N-[(3R,5S)-5-(ethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-5-methyl-1,2-oxazole-4-carboxamide
5-(1-{4-[2-(2-phenylethynyl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)-1H-1,2,3,4-tetrazole
methyl 6-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]cyclopropane-1-carboxamide
methyl 2-[(3,5-dimethylphenyl)sulfamoyl]-6-propanoyl-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-({methyl[3-(1H-pyrazol-1-yl)propyl]amino}methyl)quinolin-8-ol
1-ethyl-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-6-(propan-2-yl)pyrimidin-4-amine
5-{8-[2-(dimethylamino)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecane-2-carbonyl}pyridine-2-carbonitrile
N-[(1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}piperidin-4-yl)methyl]acetamide
5-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
4-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propanamido}-N-ethylpiperidine-1-carboxamide
(3S,5S)-1-(1-benzofuran-2-ylmethyl)-5-[(4-fluorophenyl)carbamoyl]piperidine-3-carboxylic acid
N-{[4-(dimethylamino)-1-methylpiperidin-4-yl]methyl}-4-(3-hydroxy-3-methylbutyl)benzamide
ethyl 5-[(2,6-difluorophenyl)methyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}-2-methyl-1,4-diazepan-5-one
4-methyl-3-(2-oxoimidazolidin-1-yl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]benzamide