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1-(1,3-benzoxazol-2-yl)-N-[2-(1H-pyrazol-4-yl)ethyl]piperidin-4-amine
(3S,5R)-1-(1H-imidazol-2-ylmethyl)-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
1-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-(1H-1,2,3,4-tetrazol-5-yl)piperidine
(2R)-2-amino-3-(ethylsulfanyl)-1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}propan-1-one
1-(4-{10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperazin-1-yl)ethan-1-one
5-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(4aS,7aR)-1-(3-cyclopropylpropanoyl)-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-[1-(4-propylphenyl)ethyl]acetamide
N-(3-methoxy-4-methylphenyl)-4-[(methylsulfanyl)methyl]piperidine-1-carboxamide
5-methyl-2-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine
N,3,5,7-tetramethyl-N-[1-(pyridin-2-yl)propyl]-1H-indole-2-carboxamide
(3aS,6aS)-5-(isoquinolin-5-ylmethyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N'-(3-chloro-4-fluorophenyl)-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]butanediamide
2-[1-(cyclohexylmethyl)-4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperazin-2-yl]ethan-1-ol
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1,4-diazepane
4,6-dimethyl-N-(oxan-3-ylmethyl)quinolin-2-amine
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
1-[2-(morpholin-4-yl)ethyl]-3-(2-phenyl-1,3-benzoxazol-5-yl)urea
1,9-dimethyl-4-[3-(2-oxopyrrolidin-1-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-({1-[(2-ethylpyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)thiophene-3-carboxamide
N-[3-(1H-imidazol-1-yl)propyl]-4-oxo-3,4-dihydroquinazoline-2-carboxamide
3-(2-{7-[cyclohexyl(methoxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-oxoethyl)-1,3-thiazolidine-2,4-dione
N-(1-{2-[3-(4-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-3-phenoxypropanamide
2-chloro-N-{2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}benzamide
(1S,5R)-3-(3-phenylpropyl)-6-(pyridine-3-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
3-(2,5-dihydro-1H-pyrrol-1-ylmethyl)-N-(2-methoxy-6-methylphenyl)benzamide
2-(morpholin-4-yl)-N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]pyrimidine-5-carboxamide
2-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
4-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-3-yl]benzoic acid
methyl 6-[2-(2-methoxyphenyl)acetyl]-2-[(3-methylbutyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2,2-dimethyl-3-{[(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amino}propan-1-ol
2-[2-(dimethylamino)phenyl]-5,6-dimethylpyridine-3-carbonitrile
4-methoxy-N-(2-methoxyethyl)-2-{[1-(thiophen-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-[1-(furan-3-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-(4-methoxyphenyl)-4-[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]butane-1,4-dione
2-{4-[4-(1,2-benzothiazol-3-yl)piperazine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
2-methyl-N-[3-(4-methylpiperazin-1-yl)butyl]-4-phenylpyrimidine-5-carboxamide
3-(2-methoxyphenyl)-N,N-bis(1,3-oxazol-4-ylmethyl)-1H-pyrazole-5-carboxamide
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]pyridine-3-carboxamide
8-(1H-indol-2-ylmethyl)-3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aR,7aS)-1-ethyl-4-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-3-yl}-N-[(3-methoxyphenyl)methyl]propanamide
4-(3-aminopropanoyl)-5-butyl-1-(2-methoxyphenyl)piperazin-2-one
4-(1,3-benzothiazol-2-yl)-2-[(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]phenol
2-(1-{1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-1H-1,3-benzodiazole
5-{3-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-(2,4-dimethylphenyl)-5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
2-ethoxy-5-{[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine