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4-({3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
9-(5-methylpyridine-2-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-cycloheptyl-5-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)piperidin-2-one
N-[(3-methoxyphenyl)methyl]-2,6-dimethyl-N-(2-methylpropyl)pyrimidine-4-carboxamide
(4-benzyl-1-{[3-(furan-2-yl)phenyl]methyl}piperidin-4-yl)methanol
ethyl 4-[6-(3-phenoxypropanoyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
4-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-3-yl}-2-(pyridin-4-yl)pyridine
2-methyl-4-(3-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}phenyl)butan-2-ol
(1R,3S)-7-(2H-1,3-benzodioxole-5-carbonyl)-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
(3aS,6aR)-3-[3-(4-fluorophenyl)propyl]-5-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N,4-dimethyl-2-(propan-2-yl)-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1,3-thiazole-5-carboxamide
N-[(2S)-1-{7-[(5-methyl-1,2-oxazol-3-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}-1-oxopropan-2-yl]acetamide
5-[4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenoxy]-1H-1,2,3,4-tetrazole
4-[(oxan-4-yl)sulfamoyl]-N-[(3S)-piperidin-3-yl]benzamide
N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
methyl 2-(methylsulfamoyl)-6-{2-[3-(trifluoromethyl)phenyl]acetyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-({[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
2-(4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)acetic acid
7-(2-methoxybenzoyl)-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,4-diazepane
4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
3-[methyl({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl})amino]propane-1,2-diol
(3R,4R)-4-ethyl-1-[4-methoxy-3-(morpholin-4-yl)benzoyl]piperidine-3,4-diol
2-{2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-methylphenoxy}acetamide
1-[(4-methyl-2-phenyl-1,3-thiazol-5-yl)methyl]-5-oxopyrrolidine-3-carboxylic acid
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-1-ethyl-7-methyl-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxamide
3-[1-(1H-imidazol-1-yl)butan-2-yl]-1-(6-methoxy-2H-1,3-benzodioxol-5-yl)urea
N-cyclohexyl-4-oxo-3,4-dihydroquinazoline-2-carboxamide
2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
2-[(3-fluorophenyl)methyl]-4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]morpholine
N-(1H-imidazol-2-ylmethyl)-7-(oxolan-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-(2-{5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}ethyl)-1H-1,2,3,4-tetrazole
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(4S)-3-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-4-phenyl-1,3-oxazolidin-2-one
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,6-dichlorophenyl)urea
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
8-(3-methylbut-2-enoyl)-2,8-diazaspiro[4.5]decan-3-one
2,5-dimethyl-N-{[5-methyl-2-(trifluoromethyl)furan-3-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N,3-dimethyl-4-({[1-(pyridin-3-ylmethyl)piperidin-3-yl]carbamoyl}amino)benzamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(5-propylpyrimidin-4-yl)-1,4-diazepan-5-one
5-(morpholine-2-carbonyl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
(3S,4S)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
2-(3,5-difluorophenyl)-4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
(1S,5R)-6-(2,5-dimethylfuran-3-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-{4-[(2-ethylmorpholin-4-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
N,2-dimethyl-6-(piperidin-4-yl)-N-(quinolin-2-ylmethyl)pyrimidin-4-amine
3-[3-(2-methoxyphenoxy)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[4-(3-chloro-4-fluorophenyl)piperazine-1-carbonyl]-1-methylpiperidin-4-ol