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3,5-diacetamido-N-[(4-fluorophenyl)methyl]-N-methylbenzamide
N-butyl-2-[2-(cyclopentylcarbamoyl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-[(3R,4R)-3-hydroxy-1-(oxan-4-yl)piperidin-4-yl]pyridine-3-carboxamide
N-cyclopentyl-1-[1-(2-methylpropyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
1-benzyl-5-{[3-(cyclopentylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-imidazole
N-(1-cyclopropanecarbonylazepan-3-yl)-2-(4-methyl-2-oxo-1,2-dihydroquinolin-1-yl)acetamide
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidine
2-(2-aminoethyl)-5,6-dimethyl-N-[2-(pyridin-4-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
3-(1-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}piperidin-2-yl)pyridine
N-(butan-2-yl)-N-cyclopentyl-4-acetamidobenzamide
3-[methyl({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl})amino]propanamide
4-(2-{[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]oxy}hex-5-en-1-yl)morpholine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-3-fluoro-N-methylbenzamide
3-[2-(methylsulfanyl)benzoyl]-1-(thian-4-yl)piperidine
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(trifluoromethyl)phenyl]urea
(3S,9aR)-3-benzyl-8-(2,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-amino-3-[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-[(3-methoxyphenyl)methyl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)-N-(prop-2-en-1-yl)propanamide
2-[1-(2-hydroxyethyl)-5-[2-(pyrrolidin-1-yl)-5,6,7,8-tetrahydroquinazolin-4-yl]-1H-1,2,4-triazol-3-yl]acetamide
2-(ethylamino)-N-[(4-methoxyphenyl)methyl]-N-(oxolan-2-ylmethyl)pyrimidine-5-carboxamide
N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
3-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-[2-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
1-[(1-{6-[(2-methoxyethyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
3-(1-ethoxy-2-methylpropan-2-yl)-1-(5-fluoro-2-methoxyphenyl)urea
4-cyano-N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
1-(furan-2-ylmethyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}piperidine-3-carboxamide
4-{[cycloheptyl(pyridin-3-ylmethyl)amino]methyl}-2,6-dimethoxyphenol
5-{1-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
3-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]piperidine-1-carboxamide
6-acetyl-2-amino-4-(isoquinolin-5-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}benzonitrile
N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
2-(2-oxo-2-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-2-azaspiro[4.4]nonan-3-one
1-ethyl-4-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]-1H-pyrrole-2-carbonitrile
8-(1H-indole-2-carbonyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(3-hydroxy-3-methylbutyl)-N-[(5-methoxy-1H-indol-2-yl)methyl]benzamide
4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-6-(propan-2-yl)pyrimidin-2-amine
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-methyl-1H-1,3-benzodiazole
4-{1-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-4-phenyl-1H-imidazol-5-yl}-2-ethylpyrimidine
N-cyclopropyl-1-{1-[3-(thiophen-2-yl)propanoyl]piperidin-4-yl}piperidine-3-carboxamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(pyrimidin-2-yl)-1,4-diazepan-5-one
4-(4-chloro-1-methyl-1H-pyrazole-3-amido)-N-phenylpiperidine-1-carboxamide
1-ethyl-8-[4-(1H-indol-3-yl)butan-2-yl]-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-methoxy-4-(3-methylbutanamido)phenyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
N-[(1-cyclohexylpiperidin-4-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-phenyl-1,2-oxazole-5-carboxamide
N-[1-(1-acetylpiperidin-4-yl)-1H-pyrazol-5-yl]-3-phenoxypropanamide
1-cyclopropyl-N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-5-oxopyrrolidine-3-carboxamide