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4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-[(2R)-pyrrolidine-2-carbonyl]piperidine
1-benzyl-5-(2,2-diphenylethyl)-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2S)-2-{imidazo[1,2-a]pyridin-6-ylformamido}-4-methylpentanamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-6-methyl-2-phenylpyrimidin-4-amine
2-cyclopropyl-N-(2,6-dimethylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-({5-[6-(dimethylamino)pyridin-3-yl]-4-phenyl-1H-imidazol-1-yl}methyl)-6-methyl-3,4-dihydropyrimidin-4-one
N,5-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-[(2-methoxyphenyl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
4-{1-methyl-octahydropyrrolo[1,2-a]piperazin-2-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-amine
3-{[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]pyrrolidine-3-carboxylic acid
2-(methylsulfanyl)-6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
N-methyl-N-[2-(morpholin-4-yl)ethyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
4-[2-(2-ethylphenoxy)ethyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
3-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1-methyl-1H-indole
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]acetamide
(4aS,7aR)-1-(4-ethylbenzoyl)-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(2-methoxyphenyl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-methyl-5-(propan-2-yl)-N-[2-(pyridin-3-yloxy)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-{2-[methyl(phenyl)amino]propyl}-3-phenyl-1H-pyrazole-4-carboxamide
6-[1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperidin-3-yl]pyrimidin-4-ol
N-cyclohexyl-4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carboxamide
N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-{2-[benzyl(methyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}-1,4-diazepan-5-one
1-(2-chlorophenyl)-4-[1-(methoxymethyl)cyclopropanecarbonyl]piperazine
N-[(3R,4S)-4-cyclopropyl-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-3-yl]cyclobutanecarboxamide
2-[4-(2-methoxyquinolin-3-yl)-1H-pyrazol-1-yl]acetic acid
2-(dimethylamino)-N-{2-[2-methyl-5-(morpholine-4-sulfonyl)-1H-1,3-benzodiazol-1-yl]ethyl}acetamide
1-[(3aS,6aS)-5-[3-(pyridin-3-yl)propanoyl]-octahydropyrrolo[3,4-b]pyrrol-1-yl]-3-(methylsulfanyl)propan-1-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetamide
6-methoxy-2-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(piperidin-1-yl)piperidine-4-carboxamide
3,5-dimethyl-7-[2-(4-methylphenoxymethyl)furan-3-carbonyl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine
N-[(3S,4R)-1-(3,5-difluoropyridine-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-(1H-pyrazol-1-yl)-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)propan-1-one
2-{[2-(furan-2-yl)pyrrolidin-1-yl]methyl}pyridine-3-carboxylic acid
(3R,4R)-4-ethyl-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine-3,4-diol
N-(1-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
8-(3-hydroxy-6-methylpyridin-2-yl)-2-(pyrrolidin-1-yl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(3-hydroxyphenyl)ethan-1-one
1'-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidine
methyl 4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazine-1-carboxylate
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
3-cyclohexyl-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1H-pyrazole-4-carboxamide
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-{2-[(pyridin-3-yl)amino]ethyl}urea
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(3-methyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{[1-(thiophen-2-yl)propan-2-yl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-{[5-(methylsulfanyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]methyl}cyclohexanecarboxamide
3-(azetidine-1-carbonyl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]benzene-1-sulfonamide