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2-[(2-fluorophenyl)methyl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,3-benzoxazole-6-carboxamide
N-({1-[(6,8-dimethyl-2-oxo-2H-chromen-4-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
2-(2-aminopyrimidin-5-yl)-N-[2-(dimethylamino)ethyl]-N,6,8-trimethylquinoline-4-carboxamide
3-{2-[4-(2-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
N-[7-methoxy-4-(3-methylthiophen-2-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]methanesulfonamide
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-{[(4-sulfamoylphenyl)methyl]amino}acetamide
5-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methyl-1H-1,3-benzodiazole
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-1,3-oxazolidin-2-one
2-(3-hydroxypiperidin-1-yl)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
(1S,5R)-6-(2-methoxyethyl)-3-(5-phenyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{2-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
N-{[7-fluoro-5-(quinolin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopent-1-ene-1-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
methyl 4-({[1-(cyclohexylmethyl)piperidin-3-yl]amino}methyl)benzoate
N-[2-(2-{3-[1-(dimethylamino)ethyl]phenyl}-1H-imidazol-1-yl)ethyl]acetamide
2-[4-({[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]amino}methyl)phenoxy]ethan-1-ol
(4aR,7aS)-1-benzyl-4-(2,2,3,3-tetramethylcyclopropanecarbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-ethyl-5-({2-[(3-methoxyphenyl)methyl]morpholin-4-yl}methyl)pyrimidin-2-amine
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-(4-chlorophenyl)-2-(1,3-dimethyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(1-benzyl-1H-pyrazol-3-yl)-2-[3,5-dimethyl-4-(pyridin-3-yl)-1H-pyrazol-1-yl]acetamide
methyl 4-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)benzoate
2-methoxy-3-[3-(3-methylphenyl)piperidine-1-carbonyl]pyridine
3-{1-[1-(4-acetylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
1-[(1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-2-yl)methyl]-1H-pyrazole
4-cyclobutyl-N,6-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrimidin-2-amine
3-methyl-5-[(4-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}phenyl)methyl]-4H-1,2,4-triazole
2-ethyl-N-(5-hydroxy-4,4-dimethylpentyl)pyrimidine-5-carboxamide
2-(adamantan-1-ylmethyl)-5-(dimethylamino)-2,3-dihydropyridazin-3-one
1-(2,3-dihydro-1H-inden-2-yl)-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(2-methoxyethoxy)ethan-1-one
N-(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)acetamide
N-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5-difluorobenzamide
2-[4-(1-cycloheptyl-1H-imidazol-2-yl)-2-methoxyphenoxy]acetamide
3-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-5-ethyl-1,2,4-oxadiazole
2-{[5-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)pyrimidin-2-yl](methyl)amino}acetic acid
5-(5-cyclopropyl-1,3-oxazol-4-yl)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-ethyl-1H-1,2,4-triazole
(1R,5R)-6-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(prop-2-en-1-ylsulfanyl)-N-(pyridin-3-ylmethyl)propanamide
2-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
5-[(4aR,8aR)-octahydro-2H-1,4-benzoxazine-4-carbonyl]-N-phenylpyrimidin-2-amine
4-{[(3-hydroxypropyl)[(5-methylthiophen-2-yl)methyl]amino]methyl}benzoic acid
2-[2-(1H-imidazol-1-yl)ethyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
{1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}(pyridin-2-yl)methanol
3-(2-{6-azabicyclo[3.2.1]octan-6-yl}-2-oxoethyl)-3-(4-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}-4-(1,3-thiazol-2-yl)piperazine
N,4-dimethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,3-thiadiazole-5-carboxamide
N-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
(3S,5R)-N3-[3-(dimethylamino)propyl]-N5-(4-fluorophenyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
(2E)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)-3-(pyridin-2-yl)prop-2-en-1-one