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2-(2-ethyl-1H-imidazol-1-yl)-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)acetamide
4-({ethyl[(1-methylpyrrolidin-3-yl)methyl]amino}methyl)-N-(1,3-thiazol-2-yl)benzamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}acetamide
4-(dimethyl-1,2-oxazol-4-yl)-3-(3,3,3-trifluoropropyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
4-(1H-imidazol-1-yl)-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidine-4-carboxylic acid
(1R,3S)-3-{4-[3-(4-fluorophenoxy)propyl]piperazine-1-carbonyl}cyclopentan-1-amine
2-(2-fluorophenoxymethyl)-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1,3-oxazole-4-carboxamide
3-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}acetamide
4-methoxy-N-{4-[4-(3-methoxypiperidin-1-yl)piperidin-1-yl]phenyl}benzamide
3-{[1-(propane-2-sulfonyl)pyrrolidin-3-yl]methyl}benzoic acid
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-2-(2H-1,2,3,4-tetrazol-2-yl)acetamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
4-methyl-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-1,3-oxazole-5-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
3-{ethyl[(4-methyl-1H-imidazol-5-yl)methyl]amino}-1λ6-thiolane-1,1-dione
3-[5-({4-[5-(oxan-2-yl)furan-2-yl]-1H-1,2,3-triazol-1-yl}methyl)-1,2-oxazol-3-yl]pyridine
N-methyl-4-oxo-1-(2-phenylethyl)-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
1-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-3-(1-methylpiperidin-3-yl)propan-1-one
N-(5-chloro-2-methoxyphenyl)-3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}propanamide
2-(5-phenyl-1,2-oxazole-4-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-(thiophene-2-carbonyl)piperidine
3-chloro-N-[2-(1H-imidazol-4-yl)ethyl]-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
(2S)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-methyl-2-phenylpiperazine
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N'-[2-(methylsulfanyl)phenyl]butanediamide
2-[4-(4-fluorophenyl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-1-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}ethan-1-one
4-(1-methyl-1H-pyrazol-4-yl)-2-[3-(trifluoromethyl)piperidin-1-yl]pyrimidine
(4S)-N-[(2-fluorophenyl)methyl]-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carboxamide
2-(4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
1-(2-methoxyphenyl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-4-carboxamide
1-(2-{[(2E)-3-(furan-2-yl)prop-2-en-1-yl]amino}ethyl)-N-(2-methylphenyl)-1H-1,2,3-triazole-4-carboxamide
N-[2-(2-fluorophenyl)ethyl]-3-(hydroxymethyl)-3-(2-methoxyethyl)piperidine-1-carboxamide
1-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-3-(2,4-difluorophenyl)-1-methylurea
N-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-N'-(2-ethoxyphenyl)propanediamide
1-(1-benzothiophene-5-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-(5-fluoro-2-methylbenzoyl)-4-phenoxypiperidine-4-carboxylic acid
3-methyl-4-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-2-one
N'-cyclopropyl-N-(2,5-dimethylphenyl)-N'-[(4-ethoxyphenyl)methyl]propanediamide
methyl (2S,4S)-1-methyl-4-(1H-1,2,4-triazole-5-amido)pyrrolidine-2-carboxylate
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-3-acetamidopropanamide
(1S,4S)-2-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-2-azabicyclo[2.2.1]heptane
ethyl 1-(2,6-dimethoxypyridine-3-carbonyl)-4-(3-phenylpropyl)piperidine-4-carboxylate
3,3-dimethyl-1-[(5-{[2-(propylamino)pyrimidin-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]urea
N-benzyl-2-(3-methoxypropyl)-N-methylpiperidine-1-sulfonamide
methyl 5-[2-(methylsulfanyl)-6-oxo-1,6-dihydropyrimidine-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-[4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)morpholin-2-yl]ethan-1-amine
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[3-(3-fluorophenyl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
4-cyclopentyl-2-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidine