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N-[(2,4-difluorophenyl)methyl]-3-(1H-pyrazol-1-yl)benzamide
(1R,3S)-3-[4-(benzyloxy)piperidine-1-carbonyl]cyclopentane-1-carboxylic acid
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-(3-phenylpropyl)pyrrolidine-2-carboxylate
(4aR,7aS)-1-(2-methoxyacetyl)-4-(3-methyl-1,2-oxazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[2-(dimethylamino)ethyl]-8-(5-ethyl-2-methylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-chloro-4-fluoro-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
2-cyclopropanecarbonyl-8-(9H-purin-6-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
9-(5-methyl-1H-indazole-3-carbonyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
methyl 9-(cyclopentyloxy)-7-oxo-3-(4-sulfamoylbenzoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-(cyclopropylmethoxy)-4-(1H-indazole-3-carbonyl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
N-(5-fluoro-2-oxo-2,3-dihydro-1H-indol-3-yl)-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
1-{1-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]piperidin-3-yl}-4-phenylpiperazine
4-methyl-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-4-[(3-methylphenyl)methyl]piperazine
3-(benzyloxy)-1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
5-[4-fluoro-3-(hydroxymethyl)phenyl]-N-(prop-2-en-1-yl)furan-2-carboxamide
(3aR,6aR)-2-methanesulfonyl-5-[3-(4-methylphenyl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 3-benzamido-5-[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-methoxy-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-amine
3-(piperidin-1-ylmethyl)-1-[5-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-ol
4-{4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl}-1,3-thiazol-2-amine
1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-[(dimethylamino)methyl]piperidin-3-ol
4-{[4-(prop-2-en-1-yloxy)phenyl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}({2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl})amine
1-methyl-2-oxo-8-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
3-(1-methyl-1H-1,2,3-triazol-4-yl)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}urea
7-(oxan-4-yl)-2-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
methyl 2-[(3,4-difluorophenyl)sulfamoyl]-6-(3-methylpentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(6-carbamoylpyrazin-2-yl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
1-[2-methoxy-4-({[(3-methoxyphenyl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
(1S,5R)-6-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4,5-dimethyl 1-[(3S,5S)-1-[(4-methoxyphenyl)methyl]-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
N-(2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl}ethyl)acetamide
2-[4-(4-cyanophenyl)piperazin-1-yl]-2-(5-fluoro-2-methoxyphenyl)acetic acid
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
8-(2H-1,3-benzodioxol-5-ylmethyl)-1-benzyl-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(methylsulfanyl)propyl]acetamide
2-{1-[(2-ethylpyrimidin-4-yl)methyl]azetidin-3-yl}-1H-1,3-benzodiazole
5-{1-tert-butyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}-3-chloro-1,2-dihydropyridin-2-one
3-{1-[3-(dimethylamino)benzoyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
(1S,5R)-N-(1H-indazol-7-yl)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carboxamide
N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]but-2-ynamide
1-(3-hydroxyphenyl)-4-[3-(2-methylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
6-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-benzothiazole
[7-(2-methylpyrimidin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine