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1-ethyl-N-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(2S,4S)-4-amino-N-[3-(1H-imidazol-1-yl)propyl]-1-methylpyrrolidine-2-carboxamide
3-({4-[(4-fluorophenyl)methyl]piperidin-1-yl}methyl)-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
4-methyl-7-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}sulfonyl)-3,4-dihydro-2H-1,4-benzoxazine
5-chloro-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N-(furan-3-ylmethyl)-N-methyl-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-[4-(4-fluorophenoxy)phenyl]-3-{[1-(hydroxymethyl)cyclobutyl]methyl}-3-methylurea
2-{3-[(1-methylpiperidin-4-yl)methyl]-5-{2-oxo-1-oxaspiro[4.4]nonan-4-yl}-1H-1,2,4-triazol-1-yl}acetic acid
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(2S,4R,6S)-2-ethyl-6-[4-(2-methylphenyl)phenyl]oxan-4-yl]acetamide
3-{1-[(2,4-difluoro-3-methoxyphenyl)methyl]piperidin-3-yl}propanoic acid
(1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
1-[2-(2,3-difluorophenyl)acetyl]-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
5-[(3-methylthiophen-2-yl)sulfonyl]-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-methyl-2-(2-phenyl-1H-imidazol-1-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
4-{4-[2-(2-chloro-6-fluorophenyl)acetyl]piperazin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
(1-{[2-(trifluoromethyl)pyrimidin-4-yl]amino}cyclopentyl)methanol
dimethyl(3-{[5-(1-methyl-1H-imidazol-5-yl)pyridin-2-yl]oxy}propyl)amine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(pyrimidin-4-ylmethyl)benzamide
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-(dimethyl-1,2-oxazol-4-yl)acetamide
1-{1'-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
(2S,4R)-1-benzyl-4-{[(3-chlorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
4-[(1R,2R,3S,4S)-3-aminobicyclo[2.2.1]heptane-2-carbonyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
3-chloro-N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)benzamide
1-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
5-cyclobutyl-N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1,3,4-oxadiazol-2-amine
4-(1-butyl-1H-pyrazol-4-yl)-1-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,2,3,6-tetrahydropyridine
N-ethyl-5-methyl-N-(2-methylprop-2-en-1-yl)-4-{[(6-methylpyridin-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
3-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
3-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
2-(dimethylamino)-2-(4-fluorophenyl)-N-(1-propylcyclopropyl)acetamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidine
1-(1,1-dioxo-1λ6-thiolan-3-yl)-N-[2-(furan-2-yl)ethyl]piperidine-4-carboxamide
N-(dicyclopropylmethyl)-2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(3S,4S)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
(1R,5R)-N,N-dimethyl-6-(quinoline-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
1-butyl-4-[2-(1,4-diazepan-1-yl)-2-oxo-1-phenylethyl]piperazine-2,3-dione
ethyl 4-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazine-1-carboxylate
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](ethyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
2-(1-benzofuran-2-yl)-1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-imidazole
6-(3-methylphenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
N-[3-(4,5-dihydro-1H-imidazol-2-yl)phenyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-6-one
5,6-dimethyl-3-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
1-(1H-imidazole-2-carbonyl)-4-(pyridin-3-ylmethyl)-1,4-diazepane-6-carboxylic acid
2-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carboxylic acid
2-(2-{[(1-ethylpyrrolidin-2-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid