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N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N,5-dimethyl-2-phenylfuran-3-carboxamide
2-(4-ethylpiperazin-1-yl)-N-[3-(methylsulfanyl)propyl]-2,3-dihydro-1H-indene-2-carboxamide
(4aS,8aS)-2-(1-benzyl-1H-pyrazole-4-carbonyl)-decahydroisoquinolin-4a-ol
4-{4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-2-oxopiperazin-1-yl}benzonitrile
N-[2-({5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)ethyl]acetamide
1-(5-propylpyrimidin-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]piperidin-4-amine
2-[1-(3-phenyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
N-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(oxan-4-yl)acetamide
N-[(1r,4r)-4-hydroxycyclohexyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
7-(pyridin-3-yl)-4-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl 2-({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)pyridine-3-carboxylate
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-[4-(3-methoxyphenyl)phenyl]-N,N-dimethylpiperidin-4-amine
4-chloro-5-[({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]-N,N-dimethyl-1,3-thiazol-2-amine
N-[(3-methoxyphenyl)methyl]-4-methyl-2-(methylamino)-N-(prop-2-en-1-yl)-1,3-thiazole-5-carboxamide
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N'-cyclooctyl-N-[(5-ethylpyridin-2-yl)methyl]butanediamide
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-2,3-dihydro-1H-isoindole-2-carboxamide
(3R)-3-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,2,3,4-tetrahydroisoquinoline
N,N-dimethyl-1-{2-methyl-3-[(pyridin-3-ylmethyl)amino]benzoyl}pyrrolidin-3-amine
5-{[2-(ethoxymethyl)pyrrolidin-1-yl]methyl}-1-(propan-2-yl)-1H-imidazole
2-methoxy-4-[3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carbonitrile
4-hydroxy-1-[2-(1H-indol-3-yl)acetyl]piperidine-4-carboxylic acid
2-methyl-5-(2-{2-[(6-methylpyridazin-3-yl)amino]ethyl}morpholin-4-yl)-2,3-dihydropyridazin-3-one
N2-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-5-fluoro-N4-methylpyrimidine-2,4-diamine
2-(2H-1,3-benzodioxol-5-yl)-N-[4-(pyridin-3-yloxy)phenyl]acetamide
2-chloro-5-(3,5-dimethoxyphenyl)-N-methylbenzamide
1-{2-methylthieno[3,2-d]pyrimidin-4-yl}-3-phenylpyrrolidin-3-ol
{4-[(4-chlorophenyl)methyl]-1-(3-phenylpropyl)piperidin-4-yl}methanol
(3aS,6aS)-2-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-methyl-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-1,3,4-oxadiazol-2-amine
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
4-{6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}-3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(1S,5R)-3-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 3-{[2-(3-fluorophenyl)-1,3-benzoxazol-5-yl]formamido}propanoate
1-[4-(pyridin-4-yl)piperidin-1-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
3-(3-hydroxy-3-methylbutyl)-N-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]benzamide
N-(4-methylphenyl)-3-{3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-3-oxopropanamide
2-methyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1-benzofuran-5-carboxamide
1-[(3S,4R)-1-[(6-fluoroquinolin-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
2-methyl-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]furan-3-carboxamide
3-{1-[(3-chloro-4-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-N-[(4-fluorophenyl)methyl]propanamide
2-methyl-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)oxolane-2-carboxamide
1-{[3-(4-chlorophenoxy)phenyl]methyl}-4-(pyrrolidin-3-yl)piperazine
[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl][2-(2-chlorophenoxy)ethyl]ethylamine
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-3-(1H-indol-3-yl)propan-1-one
3-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)-N-phenylpropanamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-2-methyl-N-[2-(piperidin-1-yl)ethyl]furan-3-carboxamide