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N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
N-(2-cyano-3-methylphenyl)-4-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}benzamide
1-[2-(dimethylamino)ethyl]-N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
2-amino-6-hydroxy-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-5H-indeno[1,2-b]pyridine-3-carbonitrile
1-[3-(4-chlorobenzoyl)piperidin-1-yl]-3-phenylprop-2-yn-1-one
N-ethyl-1,3-dimethyl-N-(pyridin-2-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(2-methyl-1H-imidazol-1-yl)acetyl]pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
N-[(3R,4S)-1-(carbamoylmethyl)-4-propylpyrrolidin-3-yl]-4,4,4-trifluorobutanamide
N-(2-fluorophenyl)-3-[(3-phenylpropanamido)methyl]piperidine-1-carboxamide
2-(methoxymethyl)-6-methyl-N-[2-(morpholin-4-yl)ethyl]-1-(naphthalen-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-(2-{[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)amino}ethyl)piperidin-2-one
4-[3-(2,4-difluorophenyl)propanoyl]-1-(3-methoxyphenyl)piperazin-2-one
3-(3-fluorophenyl)-N-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-4-carboxamide
3-[4-(methylamino)pyrimidin-2-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
[(4,6-dimethylpyridin-2-yl)methyl](methyl)({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)amine
N-(furan-2-ylmethyl)-N-methyl-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-chloro-2-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-5-(trifluoromethyl)pyridine
(4aS,8aR)-6-(1,3-dihydroxypropan-2-yl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
1,3-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(4-fluorophenyl)-N-(oxan-4-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
N-(diphenylmethyl)-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
ethyl 4-[4-(oxan-4-ylmethyl)-3-oxo-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl]piperidine-1-carboxylate
7-methoxy-3-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)-1,2-dihydroquinolin-2-one
[1-({1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
4-{4-[methyl(1H-pyrazol-5-ylmethyl)amino]piperidin-1-yl}-N-[(3S)-2-oxoazepan-3-yl]benzamide
3-(3-hydroxyquinoxalin-2-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)propanamide
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
1-[(2-hydroxy-3-methoxyphenyl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
6-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]pyridine-3-carbonitrile
3-[(dimethylamino)methyl]-3-hydroxy-N-[3-(2-methylphenyl)phenyl]piperidine-1-carboxamide
N-{3-[2-amino-4-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-oxopropyl}acetamide
1-(4-{[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-fluoro-4-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
4-(2,4-dimethoxyphenyl)-5,6-dimethylthieno[2,3-d]pyrimidine
1-[4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carbonyl]piperidine-4-carboxamide
5-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
2-{4-[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-N-ethylacetamide
2-methyl-5-[4-(5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
N-{3-[4-(1H-imidazol-1-ylmethyl)phenyl]phenyl}acetamide
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
1-[4-(1-ethyl-1H-pyrazole-3-carbonyl)piperazin-1-yl]-2-phenoxyethan-1-one
3-{[3-(piperidine-1-carbonyl)-1-[3-(pyridin-3-yl)propyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
(3R,4R)-1-(dimethyl-1,2-oxazole-4-carbonyl)-4-ethylpiperidine-3,4-diol
{1-[4-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-1,3-benzodiazol-2-yl}methanol
(3R,4R)-1-[(2-ethylpyrimidin-5-yl)methyl]-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
1-benzyl-4-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-1,4-diazepan-6-ol
4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-7-(2-oxoimidazolidin-1-yl)-1,2,3,4-tetrahydroquinolin-2-one
5-(1-acetylpiperidin-4-yl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N2-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-5-methylpyrimidine-2,4-diamine