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N-methyl-5-{[(oxolan-2-ylmethyl)amino]methyl}-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
(3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
N-[2-(thiophene-3-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-4-carboxamide
1-({[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]carbamoyl}methyl)piperidine-4-carboxamide
2-methoxy-2-methyl-1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]quinoxaline-5-carboxamide
N-(1-{1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
2-{4-[1-(furan-2-ylmethyl)piperidin-4-yl]piperazin-1-yl}pyridine-3-carbonitrile
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}urea
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-8-fluoroquinoline-2-carboxamide
(3S,4S)-4-methyl-1-[4-(morpholin-4-yl)benzoyl]piperidine-3,4-diol
4-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1-methyl-1H-indole
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
7-[(3-methylphenyl)methyl]-2-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decane
1-(1-benzofuran-3-carbonyl)-2-(3-methoxyphenyl)azetidine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-(furan-2-ylmethyl)-2-{3-[3-(1,3-thiazol-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
ethyl 2-{4-[3-(cyclopentylcarbamoyl)propanoyl]morpholin-3-yl}acetate
N-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
N-benzyl{[1-(pyrazin-2-yl)piperidin-4-yl]amino}sulfonamide
2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-6-(5-methylthiophen-2-yl)pyridine-3-carboxylic acid
1-cyclopropanecarbonyl-3-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]piperidine
2-ethoxy-6-{[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]methyl}phenol
2-{1-cyclopentyl-4-[(2,5-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
3-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}pyrrolidin-3-ol
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
N-(2-fluoroethyl)-3-{[1-(pyridin-3-yl)propyl]sulfamoyl}benzamide
1-[5-(pyridin-3-ylmethyl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl]butan-2-ol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-(methoxymethyl)piperidine-1-sulfonamide
N-cyclopentyl-2-(dimethylamino)-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)propanamide
4-chloro-N-(3-ethoxypropyl)-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
3-[3-(oxan-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-1H-indazole
6-(2-fluorophenyl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
1-tert-butyl-3-(cyclopropylmethyl)-5-[1-(4-methyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazole
ethyl 3-[(4-fluorophenyl)methyl]-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine-3-carboxylate
9-(4-methylpiperazine-1-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-[1-methyl-4-(quinolin-3-ylmethyl)piperazin-2-yl]ethan-1-ol
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)(4-phenylbutyl)amine
ethyl 4-[7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidine-1-carboxylate
N-[(3S,4R)-1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylpyridine-4-carboxamide
1-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-3-propylpiperidine-3-carboxylic acid
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-(1,4-dioxan-2-ylmethyl)-5-(4-methoxy-2,5-dimethylphenyl)-4-phenyl-1H-imidazole
2-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}-4-methoxyphenol
3-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-N-(pyridin-3-yl)propanamide
1-(2-{[2-(1H-indol-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}ethyl)imidazolidin-2-one