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8-cyclooctyl-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(4-chloro-2-methylphenoxy)-1-(7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
4-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1-(propan-2-yl)piperidine
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2,7-dimethylimidazo[1,2-a]pyridine-3-carboxamide
N-methyl-N-[(5-methylfuran-2-yl)methyl]-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
N'-(butan-2-yl)-N-cyclopentyl-N'-(3-phenylprop-2-yn-1-yl)butanediamide
1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-3-(4H-1,2,4-triazol-3-yl)piperidine
4-[(2,3-dimethoxyphenyl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-1,9-dioxaspiro[5.5]undecan-4-amine
3-(1H-imidazol-2-yl)-N-[1-(4-methoxyphenyl)propyl]-N-methylbenzamide
1-methyl-4-{5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}-1,4-diazepane
6-[3-(butan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
(2R,6R)-4-(4-chlorobenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-cyclohexyl-N-[1-(thian-4-yl)piperidin-4-yl]-1H-pyrazole-4-carboxamide
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
{4-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]morpholin-3-yl}methanol
5-[1-(2,3-dihydro-1H-inden-2-yl)-1H-pyrazol-3-yl]-N-(furan-3-ylmethyl)-4-methyl-1,3-thiazol-2-amine
(2S,4S)-4-({[4-(benzyloxy)phenyl]methyl}amino)-1-[(2-chlorophenyl)methyl]-N-methylpyrrolidine-2-carboxamide
N-(2-methoxyethyl)-1-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)piperidine-3-carboxamide
N-{3-[(2-ethylphenyl)carbamoyl]phenyl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,1-dioxo-3,4-dihydro-2H-1λ6,2-benzothiazine-3-carboxamide
N-{1-[7-(2H-1,3-benzodioxole-5-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}furan-3-carboxamide
(2S,3S)-2-amino-1-{4-[(4-cyclohexyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-3-methylpentan-1-one
N-[4-(3-methoxyphenyl)phenyl]-1-[2-(1H-pyrazol-1-yl)acetyl]pyrrolidine-2-carboxamide
(3S,4R)-4-(3-fluorophenyl)-1-(3-methyloxetane-3-carbonyl)pyrrolidine-3-carboxylic acid
2-(2-methoxyphenyl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}benzenesulfonamide
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-(1-methyl-1H-imidazol-2-yl)piperidine
3,5-dichloro-N-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-4-methylbenzamide
3-methyl-8-(2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1-methyl-1H-imidazole-5-carbonyl)pyrrolidin-3-yl]pyridine-2-carboxamide
N-[(2-methylphenyl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-(2-chloro-3,5-difluorophenyl)-3-(2-ethyl-2,5-dihydroxypentyl)urea
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(1H-pyrazol-1-ylmethyl)piperidine
1-(propan-2-yl)-N-[1-(thian-4-yl)piperidin-4-yl]-1H-pyrazole-4-carboxamide
7-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)-2,7-diazaspiro[4.5]decane
1-[7-(5-methylthiophen-2-yl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
1-methyl-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
2-ethyl-N-[1-(furan-2-carbonyl)piperidin-3-yl]pyrimidine-5-carboxamide
[9-(3-fluorobenzoyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
N-phenyl-5-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine-1-carbonyl}pyrimidin-2-amine
6-[(diethylamino)methyl]-N-(1-phenylethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]pyridine-3-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(2,3,4-trifluorophenyl)ethan-1-one
4-(ethanesulfonyl)-2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]phenol
ethyl 1-(1H-1,3-benzodiazole-5-carbonyl)-3-[(3-chlorophenyl)methyl]piperidine-3-carboxylate
4-{2-[(4-methylphenyl)sulfanyl]propyl}-1λ6-thiomorpholine-1,1-dione
2-{4-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1H-pyrazol-1-yl}-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
4-(8-methoxyquinolin-5-yl)-2-(1,2-oxazol-5-yl)phenol