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(1R,2S)-2-[1-(2-hydroxyethyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-N-methylcyclohexane-1-carboxamide
1-(3-chlorophenyl)-4-(2-methoxy-2-phenylacetyl)piperazin-2-one
N-[(3S,4R)-1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
ethyl 1-{[4-(2-oxoimidazolidin-1-yl)phenyl]methyl}-3-(2-phenoxyethyl)piperidine-3-carboxylate
5-ethyl-3-(1-hydroxypropan-2-yl)-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-(3-chlorobenzoyl)-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
2-amino-6-(3-hydroxyphenyl)-4-[2-(pyrrolidin-1-yl)pyrimidin-5-yl]pyridine-3-carbonitrile
N-ethyl-5-methyl-4-(4-methylpiperazin-1-yl)-N-(2-methylprop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
N-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-4-methanesulfonylpiperazine-1-carboxamide
5,6-dimethyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-oxo-1,2-dihydropyridine-3-carboxamide
[(3,4-dimethoxyphenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
2-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidine-1-carbonyl]pyridin-3-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]piperidin-3-ol
4-[1-(3-chlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1,2,3-thiadiazole
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]acetamide
1-({1-[(2-chloro-6-fluorophenyl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl}methyl)-1H-1,2,3,4-tetrazole
N-[2-(furan-2-yl)ethyl]-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
1-[1-(2-aminoacetyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
4-(ethylamino)-N-(2-methoxyethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
9-(but-3-yn-1-yloxy)-4-(2,5-dimethoxybenzoyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-cyclopentyl-5-oxo-N-[(4-phenyloxan-4-yl)methyl]pyrrolidine-3-carboxamide
N-(oxolan-2-ylmethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
2-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-(2-methoxyacetyl)-N-[phenyl(pyridin-4-yl)methyl]piperidine-4-carboxamide
(2S,4R)-4-amino-N-methyl-1-(naphthalene-1-carbonyl)pyrrolidine-2-carboxamide
5'-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3',5',6',7'-tetrahydrospiro[cyclohexane-1,4'-imidazo[4,5-c]pyridine]
N-[2-(1H-imidazol-2-yl)ethyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(4-chloro-2-fluorophenyl)-1-[(2S)-oxolan-2-ylmethyl]-1H-imidazole
2-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-N-(2-methylbutan-2-yl)-2-oxoacetamide
1-{2-[(4aS,7aR)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethyl}-3,3-dimethylurea
2-(adamantan-1-yl)-5-{2-azaspiro[4.4]nonane-2-carbonyl}pyrimidin-4-ol
5-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}-2-methyl-3,4-dihydropyrimidin-4-one
4-(benzyloxy)-1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
2,4-dimethoxy-6-[3-(pentan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrimidine
[1-(1-benzofuran-2-ylmethyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
4-methylphenyl (7S,9aR)-7-(1H-indol-3-ylmethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
N,5-diethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1,3-oxazole-4-carboxamide
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(pyridin-4-ylmethyl)amine
(1R,5R)-6-(5-methoxyfuran-2-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
4-[({[4-(butan-2-yloxy)-3-chlorophenyl]methyl}amino)methyl]-1,3-thiazol-2-amine
N-[2-(3-phenylpiperidin-1-yl)ethyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2,5-dimethyl-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]furan-3-carboxamide
2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-benzoxazole
(1S,5R)-3-(propane-1-sulfonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(4-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1-methylpiperazin-2-yl)methanol
N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-methyl-3-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
methyl 9-(cyclopentyloxy)-7-oxo-3-[4-(2-oxopyrrolidin-1-yl)benzoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[5-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
2-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-6-(4-methylpiperazine-1-carbonyl)pyrazine