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5-(azepan-1-yl)-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole
2-(1-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)pyridine
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-(trimethyl-1H-pyrazol-1-yl)acetamide
6-oxo-N-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}-1,6-dihydropyridine-3-carboxamide
5-[3-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
(4aR,7aS)-1-ethyl-4-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[3-(1H-pyrazol-1-yl)propanoyl]pyrrolidin-3-yl]acetamide
5-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
6-methyl-2-({4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)quinolin-4-ol
2-butyl-N-(quinolin-6-ylmethyl)-1,3-benzoxazole-5-carboxamide
2-amino-6-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-4-(pyridin-3-yl)pyridine-3-carbonitrile
8-(3-methyl-1H-pyrazole-5-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-(azepane-1-carbonyl)-N-cyclohexyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
1-cyclopentyl-4-{[(pyrimidin-2-yl)amino]methyl}pyrrolidin-2-one
N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}acetamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
1-(1-{[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}cyclohexyl)piperidine
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(2-methylpyrimidin-5-yl)methyl]piperidin-4-ol
(1R,5R)-3-(pyridine-2-carbonyl)-6-(3,3,4,4-tetrafluorobutyl)-3,6-diazabicyclo[3.2.2]nonane
3-{2-oxo-2-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethyl}imidazolidine-2,4-dione
8-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
1-{3-[2-(methylcarbamoyl)ethyl]phenyl}-5-oxopyrrolidine-3-carboxylic acid
9-(2,5-dimethylfuran-3-carbonyl)-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-(5-phenyl-1H-indazol-1-yl)acetamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(2-methylpyrimidin-5-yl)methyl]piperidine-4-carboxamide
2-(5-{[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]methyl}furan-2-yl)benzonitrile
(4aS,8aR)-1-(2-methylpropyl)-6-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(4-methylphenoxy)acetamide
(2E)-1-[(4aR,8aS)-6-(oxane-4-carbonyl)-decahydro-1,6-naphthyridin-1-yl]-3-(4-fluorophenyl)prop-2-en-1-one
N-[2-(2-ethyl-1,3-thiazol-4-yl)ethyl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
1-(2-cyclopentaneamido-5-methylphenyl)-5-oxopyrrolidine-3-carboxylic acid
2-methoxy-1-(1'-{[1-(propan-2-yl)piperidin-4-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
5-(4-methyl-1H-imidazol-2-yl)-3-(2-phenylethyl)-1,2,4-oxadiazole
3-{2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
2-{4-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1H-1,2,3-triazol-1-yl}-N,N-diethylacetamide
4-[1-(4-{5-[(4-methylpiperazin-1-yl)methyl]pyridin-2-yl}phenyl)ethyl]morpholine
5-chloro-3-{1-[(4-fluorophenyl)methyl]-3-methyl-1H-1,2,4-triazol-5-yl}-4,6-dimethyl-1,2-dihydropyridin-2-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(cyclohexylmethyl)-6-oxopiperidine-3-carboxamide
2-(dimethylamino)-N-[(2-methylphenyl)methyl]-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
N-{1-[1-(2,5-dimethylpyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
N-(1-carbamoylcyclopentyl)-6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-(piperidin-3-ylmethyl)-N-[2-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-ethyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
8-(8-methoxyquinolin-2-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(1-cycloheptylpiperidin-3-yl)-8-methylimidazo[1,2-a]pyridine-2-carboxamide
4-(2-ethoxybenzoyl)-1-methylpiperazine-2-carboxylic acid
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-(5-propyl-1,3,4-oxadiazol-2-yl)-3-oxa-9-azaspiro[5.5]undecane
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-(2-methylphenyl)-1,4-diazepane-1-carboxamide