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2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-4-oxo-N-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
8-(2-benzyl-1,3-thiazole-4-carbonyl)-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclopentyl-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(4aS,8aR)-6-(2,5-dimethylfuran-3-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
(4aR,7aS)-1-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-3-(pyrrolidin-1-yl)propanamide
N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-(1-cyclopentyl-1H-pyrazol-5-yl)urea
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(2,2,2-trifluoroethyl)propanamide
2-{4-[4-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}pyrimidine
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)morpholine-4-sulfonamide
(2S,4S)-4-[2-(4-chlorophenyl)acetamido]-N-(furan-3-ylmethyl)-N,1-dimethylpyrrolidine-2-carboxamide
1-[1-(4-methoxy-3,5-dimethylbenzoyl)azetidin-3-yl]-2-methylpiperidine
2-fluoro-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-5-sulfamoylbenzamide
2-(adamantan-1-yl)-4-hydroxy-N-(2-methoxy-2-methylpropyl)pyrimidine-5-carboxamide
4-[(1H-1,3-benzodiazol-2-ylmethyl)amino]-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
4-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]ethan-1-one
5-{1-[(3-chloro-1H-indol-2-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
(1S,6R)-3-[3-(piperidine-1-carbonyl)pyridin-2-yl]-3,9-diazabicyclo[4.2.1]nonane
3-(carbamoylmethoxy)-N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]benzamide
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-2-(pyridin-3-yl)pyridine
6-methyl-2-phenyl-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}pyrimidin-4-amine
2-(2-{1-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrrol-1-yl)pyridine
8-(cyclopropylmethyl)-N-(2,6-dimethylphenyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-chloro-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}pyridine-4-carboxamide
2-(2-methoxyethyl)-9-(2-methyl-2-phenylpropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-carboxylic acid
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(2-hydroxyphenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(4-{[(2-chlorophenyl)methyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
4-{1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}-2,1,3-benzoxadiazole
N-methyl-N-propyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-cyclobutanecarbonyl-4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-1,4-diazepane
3-{[(2-methyl-1H-imidazol-4-yl)methyl][(5-methylthiophen-2-yl)methyl]amino}propan-1-ol
1-[1-(hydroxymethyl)-9-propyl-3,9-diazaspiro[5.5]undecan-3-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
4-(1-ethyl-1H-imidazol-2-yl)-1-[2-(4-fluorophenoxy)ethyl]piperidine
3-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}phenol
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-chlorobenzamide
3-[(2,6-difluoro-3-methylphenyl)methyl]-9-methyl-3,9-diazaspiro[5.6]dodecan-10-one
1-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
1-(3-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-3-oxopropyl)piperidin-2-one
ethyl 5-[(3-methylquinoxalin-2-yl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
8-(1-benzofuran-2-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-ethyl-8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-({2-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-[ethyl(propyl)amino]-2-(4-fluoro-3-methylphenyl)acetic acid
5-(morpholine-4-sulfonyl)-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline
3-{5-[1-(oxan-4-yl)piperidine-4-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
1-(3-methoxyphenyl)-4-[3-(2-methoxyphenyl)propanoyl]piperazin-2-one