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2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[3-(1,3-oxazol-5-yl)phenyl]acetamide
2-(1-benzothiophen-2-ylmethyl)-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-N-(oxan-4-yl)piperidin-4-amine
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-3-oxo-3,4-dihydroquinoxaline-2-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[5-(methoxymethyl)furan-2-carbonyl]piperidine-4-carboxylate
2-(2-methoxyethyl)-8-[3-(1H-pyrazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(2-chloro-4-fluorophenoxymethyl)-N-(3-hydroxypropyl)-N-methyl-1,3-oxazole-4-carboxamide
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine
1-cyclopropyl-4-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]pyrrolidin-2-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-(2-oxopiperidin-1-yl)butanamide
2-(4-methylphenyl)-5-[2-(1,3-thiazol-2-yl)piperidine-1-carbonyl]pyrimidin-4-ol
1-(4-benzylpiperidin-1-yl)-3-[1-(2-hydroxyacetyl)piperidin-4-yl]propan-1-one
5-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]pyrazine-2-carboxamide
methyl 6-(2-oxo-2-phenylacetyl)-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2,3-dimethoxybenzamide
3-benzyl-8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-methylphenyl)-5-[({[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amino)methyl]-1,3-thiazol-2-amine
{[3-(2,4-dimethoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
2-(2,5-dioxoimidazolidin-1-yl)-N-[3-(4-ethoxyphenyl)propyl]acetamide
2-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-1,3-benzothiazole
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-4-(pyridin-2-yl)pyrimidin-2-amine
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
(3R,4S)-4-phenyl-1-[4-(piperidin-1-yl)benzoyl]pyrrolidin-3-amine
N-[5-(2-chloro-4-fluorophenyl)pyridin-2-yl]methanesulfonamide
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-methyl-N-(propan-2-yl)propanamide
2-[2-(4-methanesulfonylphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
3-[(2-methoxypyrimidin-5-yl)methyl]-3,9-diazaspiro[5.6]dodecan-10-one
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
3-(4-hydroxyphenyl)-N-(2-methoxyethyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
N-[2-(naphthalen-2-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-methyl-1-(4-methylphenyl)-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperazin-2-one
3-amino-1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propan-1-one
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-{imidazo[1,2-b]pyridazin-6-yl}piperazine
3-(2-methyl-1H-1,3-benzodiazol-6-yl)-1-(2,2,6,6-tetramethylpiperidin-4-yl)urea
1-{1-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
8-(2-acetylbenzoyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
9-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-(quinolin-4-ylmethyl)benzamide
4-(4-fluorophenyl)-N-(1-methyl-2-oxopyrrolidin-3-yl)benzamide
1-[4-(2-chlorophenyl)piperazin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)amine
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
(1S,5R)-3-(4-chloro-3-fluorobenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
3-({[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
1-[(3-chloro-2,6-difluorophenyl)methyl]-2-(2-methoxyethyl)piperidine
N-(2-phenoxyethyl)morpholine-2-carboxamide
1-(2-amino-6-methylpyrimidin-4-yl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-(2-aminoethyl)-4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxybenzamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide