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6-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-phenylimidazo[1,2-a]pyridine
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-(1,3-thiazol-2-ylmethyl)benzamide
1-(2-methylpyridin-4-yl)-1H-1,3-benzodiazole
N-[(1-cyclopentylpiperidin-4-yl)methyl]-6-oxo-N-(pyridin-3-ylmethyl)-1,6-dihydropyridine-2-carboxamide
N-ethyl-N-(4-hydroxybutyl)-3-(5-methylfuran-2-yl)benzamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-[2-(6-hydroxy-1,4-diazepan-1-yl)-2-oxoethyl]-2,3-dihydro-1H-indazol-3-one
[5-(4-aminophenyl)-1H-1,3-benzodiazol-2-yl]methanol
3-{1-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}benzonitrile
2-methoxy-5-({3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)phenol
1-(4-{2-[2-(3-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2,3-dimethyl-7-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}-1H-indole
(2S)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,3-dihydro-1H-indole-2-carboxamide
2-{1-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}-5-ethylpyridine
4-(5-tert-butyl-1H-pyrazol-3-yl)-1-methyl-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-6-fluoroquinolin-4-ol
3-{2-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
4-({[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl]amino}methyl)benzene-1-sulfonamide
2-methyl-6-{1-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}pyrimidin-4-ol
[1-(2-{[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]amino}ethyl)piperidin-2-yl]methanol
5-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2-carbonitrile
2-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-2-yl)pyridine
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]propan-1-one
3-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-[2-(ethylsulfanyl)phenyl]urea
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
N-cyclohexyl-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-4-yl]propanamide
5-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1,3-oxazole-4-carboxamide
2-(4-{[4-(methylsulfamoyl)phenyl]methyl}morpholin-3-yl)acetic acid
2-ethoxy-1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]ethan-1-one
N-ethyl-8-methoxy-N-(pyridin-4-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(1R,5S)-N-(2-chloro-4-fluoro-5-methylphenyl)-6-azabicyclo[3.2.1]octane-6-carboxamide
1-{4-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]phenyl}-1H-1,2,4-triazole
(1S,2S,4R)-1,7,7-trimethyl-4-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}bicyclo[2.2.1]heptan-2-ol
2-(butylsulfanyl)-5-[(3-methoxypiperidin-1-yl)methyl]pyrimidine
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl)[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]amine
1-(3-methoxyphenyl)-4-{[4-(propan-2-yloxy)phenyl]methyl}piperazin-2-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrrolidin-3-yl]pyridine-4-carboxamide
6-(benzyloxy)-4-(1-ethyl-1H-pyrazole-4-carbonyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
N-{4-[(benzyloxy)methyl]-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl}methanesulfonamide
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(1,3-thiazole-4-carbonyl)-1,4-diazepan-2-one
(3R,5S)-N-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]-5-(piperidine-1-carbonyl)piperidine-3-carboxamide
4-ethyl-3-(4-hydroxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4,6-dimethyl-2-oxo-N-[2-(4-sulfamoylphenyl)ethyl]-1,2-dihydropyridine-3-carboxamide
1-(2-methoxyphenyl)-4-(2-methyl-2-phenylpropanoyl)piperazin-2-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]piperidin-3-ol