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N-(1-{1-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-methylbutanamide
(4aR,7aS)-1-(2-methylpropyl)-4-[5-(propan-2-yl)thiophene-3-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(5-methyl-1,2-oxazole-3-carbonyl)-3-[2-(2-methylphenyl)ethyl]piperidine
4-methyl-N-{2-[4-(quinolin-4-yl)-1H-1,2,3-triazol-1-yl]ethyl}pyridin-2-amine
ethyl 3-[(2-methylphenyl)methyl]-1-(prop-2-ene-1-sulfonyl)piperidine-3-carboxylate
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)propyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-(benzyloxy)-1-(dimethyl-1,2-oxazole-4-carbonyl)piperidine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylpyridine-2-carboxamide
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[3-(propan-2-yloxy)propyl]propanamide
4,4,4-trifluoro-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]butanamide
5-[(benzyloxy)methyl]-1-ethyl-3-(oxolan-3-yl)-1H-1,2,4-triazole
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-5-hydroxypyrazine-2-carboxamide
N-[(1R,3R)-3-aminocyclopentyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-(4-{octahydropyrrolo[1,2-a]piperazin-2-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-yl)pyridine
2-{4-[5-(2-methylphenyl)-4-(4-methylphenyl)pyrimidin-2-yl]piperazin-1-yl}ethan-1-ol
methyl 4-[5-(2-fluoro-5-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]butanoate
1-(3-fluoro-4-methylphenyl)-3-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}urea
5-{3,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
methyl (2S,4R)-1-benzyl-4-(2-phenylquinoline-4-amido)pyrrolidine-2-carboxylate
4-(1-benzofuran-2-ylmethyl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
N-[(6-methylquinolin-5-yl)methyl]-3-(pyridin-3-yl)propanamide
(5-{1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1H-imidazol-2-yl}furan-2-yl)methanol
5-(2-fluoro-6-methoxyphenyl)pyrimidine
2-[(4-chlorophenyl)methyl]-N-[2-(3-methylpyridin-2-yl)ethyl]-1,3-benzoxazole-5-carboxamide
4-[3-(benzyloxy)propyl]-6-methylpyrimidin-2-amine
(4aS,7aR)-1-[(2,3-dimethoxyphenyl)methyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4S)-1-[(3-cyanophenyl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
1-ethyl-N-(2-hydroxyethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)-N-[3-(methylsulfanyl)phenyl]piperidine-1-carboxamide
2-[(4-methoxyphenyl)methyl]-4-(thian-4-yl)morpholine
(2S,4S)-N-(2-phenylethyl)-1-[(2E)-3-phenylprop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
(1R,3S)-7-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-methoxy-7-azaspiro[3.5]nonan-1-ol
1-(cyclohexylmethyl)-3-[(diethylamino)methyl]-3-hydroxypiperidin-2-one
5-fluoro-2-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}pyrimidine
1-(carbamoylmethyl)-N-methyl-N-[2-(phenylsulfanyl)ethyl]piperidine-3-carboxamide
2-{3,5-dimethyl-4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamido]-1H-pyrazol-1-yl}acetic acid
2-methoxy-5-{[2-methyl-4-(3-methylphenyl)-5-oxopiperazin-1-yl]methyl}benzoic acid
7-methyl-3-(piperidin-1-ylmethyl)-1,2-dihydroquinolin-2-one
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
1-{3-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-5-(dimethylsulfamoyl)benzoyl}piperidine-3-carboxamide
N-(3-methoxypropyl)-N-methyl-3-[(2-propyl-2,5-dihydro-1H-pyrrol-1-yl)sulfonyl]benzamide
2-[(2-fluorophenyl)methyl]-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,3-benzoxazole-6-carboxamide
3-{5-[1-(2-methyl-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
3-(2,3-dimethylphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
3-(2-chlorophenyl)-N-(2-acetamidoethyl)-3-phenylpropanamide
1-[(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(dimethylamino)propan-1-one
3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
1-[(4-ethylphenyl)methyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-cyclopropyl-3,5-dimethyl-N-{[4-(methylsulfanyl)phenyl]methyl}-1H-pyrazole-4-carboxamide