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2-(azepan-1-yl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
1-(2-ethoxyethyl)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-[(3-chlorophenyl)methyl]-5-[(3-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
3-{[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-indazole
(1S,5R)-3-methyl-6-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
(2R,6R)-4-[(2,3-dimethoxyphenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(4aS,8aR)-6-[3-(benzylsulfanyl)propanoyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-(1-benzylpyrrolidin-3-yl)-3-{1-[3-(1H-pyrazol-4-yl)propanoyl]piperidin-4-yl}propanamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-6-methoxy-N,3-dimethyl-1-benzofuran-2-carboxamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[2-(pyridin-3-yl)ethyl]acetamide
7-(2-methylphenyl)-4-(1H-pyrrole-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-yl]methyl}pyridine-3-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
methyl 3-(oxolane-3-amido)-1-(3-phenylpropyl)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-2-(2-methyl-1H-imidazol-1-yl)propan-1-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1H-1,2,3-benzotriazole-5-carboxamide
N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]oxane-2-carboxamide
4-{[1-(2-chlorophenyl)piperidin-4-yl]amino}-N,N-dimethylbutanamide
N-[2-(dimethylsulfamoyl)ethyl]-5-(3-methoxyphenyl)furan-2-carboxamide
4-[3-(2-benzyl-5-oxopyrrolidin-2-yl)propanoyl]-1-[(3-fluorophenyl)methyl]piperazin-2-one
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-(quinolin-3-ylmethyl)acetamide
N-[(4-chlorophenyl)(pyridin-3-yl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
4-[(4-ethoxy-3-methoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(3-{[methyl(quinolin-5-ylmethyl)amino]methyl}phenoxy)ethan-1-ol
8-[2-(2-hydroxyethyl)-3-oxopiperazine-1-carbonyl]-2-methyl-1,4-dihydroquinolin-4-one
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]piperidine-3-carboxamide
N-[(4-fluorophenyl)methyl]-N-(1-hydroxybutan-2-yl)-4-oxopentanamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
(4aS,8aR)-6-[(3-fluorophenyl)methyl]-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
1-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-4-(1H-imidazol-2-yl)-1H-1,2,3-triazole
(2R,4S)-4-hydroxy-1-(quinolin-8-ylmethyl)piperidine-2-carboxylic acid
1-[(2-fluoro-4-methoxyphenyl)methyl]-2-(methoxymethyl)piperidine
(1R,3S)-7-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
N-[3-(dimethylamino)phenyl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-2-ylmethyl)piperidin-3-yl]propanamide
N-(2-methoxyethyl)-2-[(2R)-oxolane-2-carbonyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2,6-dimethyl-4-{2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidine-1-carbonyl}quinoline
1-methyl-4-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrrolidin-2-one
1-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-3-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
4-({1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperidin-4-yl}methyl)morpholine
N-{1-[(4-chlorophenyl)methyl]cyclopropyl}-1-(2-methoxyacetyl)piperidine-4-carboxamide
N-{[1-(dimethylsulfamoyl)piperidin-3-yl]methyl}-2,3-dimethoxybenzamide
N,N-dimethyl-1-(5-methyl-4-{[(5-methylfuran-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)pyrrolidin-3-amine
(4aS,7aR)-1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-({3-methoxy-4-[4-(trifluoromethyl)phenoxy]phenyl}methyl)pyrrolidine
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-2-ethylpyrimidine
N-({1-[3-(1H-pyrazol-1-yl)propanoyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
methyl 4-{2-[(2-chlorophenyl)methyl]morpholine-4-carbonyl}benzoate