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N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-4-methyl-1H-imidazole-2-carboxamide
(3S,4R)-3-benzyl-4-methyl-1-(3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-ol
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidin-3-yl]propanoic acid
1-[(2-fluorophenyl)methyl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
2-[2-(dimethylamino)ethyl]-9-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-2-{5-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}butanamide
2-methoxy-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-(3-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}propyl)morpholine
1-[2,2-dimethyl-1-(thiophen-2-yl)cyclopropanecarbonyl]-4-(pyrrolidine-1-carbonyl)piperidine
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
3-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-ol
4-hydroxy-1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}piperidine-4-carboxylic acid
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
1-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-3-(prop-2-en-1-yl)urea
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)piperidine
2-acetyl-8-(3-fluoro-4-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-methyl-4-(4-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}phenyl)but-3-yn-2-ol
(1S,3R)-3-amino-N-(2,2-diphenylpropyl)cyclopentane-1-carboxamide
3-(2-methyl-1H-imidazol-1-yl)-N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]propanamide
2-methyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-5-sulfamoylbenzamide
(4aS,7aR)-1-[(6-methylpyridin-2-yl)methyl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-[2-(oxan-4-yl)ethyl]acetamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(oxolan-3-ylmethyl)piperidine-4-carboxamide
{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}(thiophen-2-yl)methanol
[(3R,4R)-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-({1-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)cyclohexanecarboxamide
N-{2-[2-(methylcarbamoyl)ethyl]phenyl}-4-(4-methylphenyl)piperazine-1-carboxamide
2-(2-methoxyethyl)-8-[(2-propoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-benzyl-8-(5-oxo-2,5-dihydro-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(1-ethyl-1H-pyrazol-3-yl)methyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
N-({1-[(3-chlorophenyl)methyl]piperidin-3-yl}methyl)-3-phenylpropanamide
7-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
dimethyl(2-{2-[1-(quinoline-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
N-[(3R,4R)-1-(3-cyano-4,6-dimethylpyridin-2-yl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
1-(2-phenylethyl)piperidin-3-amine
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-{[(3-methylphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(4-methoxyphenyl)-N-methylcyclopentane-1-carboxamide
1,3-dimethyl-2,6-dioxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(5-methylpyridine-2-carbonyl)pyrrolidine-3-carboxylic acid
2-[(6-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyrimidin-4-yl)amino]ethan-1-ol
3-methyl-5-{[3-(thiophen-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2-benzoxazole
{[2-(2-methylphenoxy)pyridin-3-yl]methyl}(pyridin-2-ylmethyl)amine
(3aR,6aR)-2-methyl-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
7-(3-chlorophenyl)-4-(furan-3-carbonyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
5,6-dimethyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}pyrimidin-4-amine
1-[3-(2-methoxyethyl)-5-[4-(piperidin-1-yl)phenyl]-1H-1,2,4-triazol-1-yl]butan-2-ol
9-[(4-chlorophenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(1,3-benzothiazol-2-yl)-4-(5-methyl-1,2,4-oxadiazol-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-ethyl-3-{[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one