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5,6-dimethyl-3-[4-(thiophene-2-carbonyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
(3S,4S)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
9-(5-ethyl-1H-pyrrole-2-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(5-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)-N-(2-hydroxyethyl)propanamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}propanamide
N-{2-[1-(7-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)piperidin-2-yl]ethyl}acetamide
1-(cyclohexylmethyl)-5-(1H-imidazol-4-ylmethyl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
N-cyclopentyl-1-{1-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
4-{1-[3-(2-phenylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}pyridine
3-(3-fluorophenyl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)propanamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[3-(methylsulfanyl)propyl]benzamide
5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-(1-methyl-1H-pyrazol-4-yl)pyridine
8-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
1-(3,4-dimethylphenyl)-N-(isoquinolin-5-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[(1S,5R)-6-[3-(morpholin-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-3-(2-methylphenyl)piperidine
(2S)-2-amino-1-{4-[benzyl(methyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-3-hydroxypropan-1-one
(3R,4S)-1-(1,3-benzothiazol-2-yl)-4-propylpyrrolidin-3-amine
(4aS,8aR)-6-(1-aminocyclopropanecarbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
(4aR,8aS)-6-{[5-(2-chlorophenyl)furan-2-yl]methyl}-1-[2-(3-methoxyphenyl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-{1-[2-(3-methoxyphenyl)ethyl]-1H-imidazol-2-yl}phenol
7-(cyclohexylmethyl)-2-methyl-2,7-diazaspiro[4.5]decan-6-one
1-(4-acetylphenyl)-3-{[4-(hydroxymethyl)oxan-4-yl]methyl}-3-methylurea
4-(2-fluorophenoxy)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
{5-[1-(cyclohexylmethyl)-3-methyl-1H-1,2,4-triazol-5-yl]furan-2-yl}methanol
2-(2-cyclopropylpyrimidin-5-yl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)quinoline-4-carboxamide
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
4-{2-[(3-methoxyphenyl)carbamoyl]ethyl}-N-[2-(methylsulfanyl)phenyl]piperidine-1-carboxamide
N,N-dimethyl-5-({methyl[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amino}methyl)-1,3-thiazol-2-amine
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
N-butyl-4-chloro-1-methyl-N-(pyridin-4-ylmethyl)-1H-indole-2-carboxamide
5-methyl-1'-{[3-(5-methylfuran-2-yl)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-4-(2-propoxyethyl)piperazine
3-methyl-1-{1-[6-(pyridin-3-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
3-{[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]sulfonyl}benzonitrile
2-[(dimethylcarbamoyl)amino]-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-2-(pyridin-3-yl)-N-(pyridin-3-ylmethyl)acetamide
methyl 2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]pyridine-3-carboxylate
N4-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-6-(morpholin-4-yl)pyrimidine-2,4-diamine
N-[2-(3-methoxyphenyl)ethyl]-5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
(2S,4R)-4-amino-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpyrrolidine-2-carboxamide
2-{[4-(2-methoxy-5-methylphenyl)-5-(1-methyl-1H-pyrazol-3-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-{[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)pyrrolidin-3-yl]methyl}benzamide
4-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}morpholine
3-hydroxy-3-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)-1-(2-phenylethyl)piperidin-2-one
(3S,4S)-1-(4-methyl-1H-imidazole-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
1-cyclobutanecarbonyl-4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1,4-diazepane
4-[2-(2,4-dichlorophenoxy)acetamido]oxane-4-carboxylic acid
1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-4-amine
methyl (2S,4S)-1-[1-(2-phenylethyl)piperidin-4-yl]-4-[2-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate