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5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(1-methylpyrrolidin-3-yl)pyridin-2-amine
3-[2-(3,4-difluorophenyl)ethyl]-1-(oxane-4-carbonyl)piperidine
[(4-fluoro-3-methoxyphenyl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
2-(1-cyclohexyl-4-{6-[ethyl(methyl)amino]pyrimidin-4-yl}piperazin-2-yl)ethan-1-ol
4-(2-methyl-1H-imidazol-1-yl)-1-[2-(pyridin-2-yl)acetyl]piperidine-4-carboxylic acid
1-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-4-(pyridin-3-yl)piperidin-4-ol
N-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-2-(pyridin-3-yl)piperidine-1-carboxamide
(5S,9aS,9bS)-5-(2-fluorophenyl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
ethyl 4-{2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetyl}piperazine-1-carboxylate
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({imidazo[1,2-a]pyrimidin-2-ylmethyl})amine
3-[2-(dimethyl-1,3-thiazol-4-yl)-N-methylacetamido]-N-methylbutanamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(furan-3-ylmethyl)piperidine-4-carboxamide
(7S,9aR)-N-cyclohexyl-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-cyclopropyl-3-{5-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
5,6,7-trimethoxy-N,N-dimethyl-3-{[(propan-2-yl)amino]methyl}quinolin-2-amine
1-methyl-4-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[2-(piperidin-1-ylmethyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
2-(4,6-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
N-[3-(1H-imidazol-1-yl)propyl]-4-methyl-2-(4-methylpiperazin-1-yl)pyrimidine-5-carboxamide
N-(2-{[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}ethyl)-N-methylmethanesulfonamide
(4aR,7aS)-1-{2-[(2,2-dimethylpropyl)(methyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(ethoxymethyl)-N-(thiolan-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(1,3-benzothiazol-2-yl)-3-{[(1-carbamoylethyl)(methyl)amino]methyl}benzamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-(quinolin-6-ylmethyl)-1H-pyrazole-4-carboxamide
2-{[(1R,5S,6S)-6-{[2-(dimethylamino)ethyl](ethyl)carbamoyl}-3-azabicyclo[3.1.0]hexan-3-yl]methyl}benzoic acid
N-[(4-methylphenyl)(pyridin-4-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
4-(4-chlorophenyl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)butanamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(2-methoxyethyl)-5-(methoxymethyl)-N-methyl-1H-pyrazole-4-carboxamide
2-(2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-1H-pyrrol-1-yl)pyrimidine
2-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)acetamide
3-{[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydro-1,2,3-benzotriazin-4-one
N-[1-(4-methoxyphenyl)ethyl]-N,2-dimethyl-2-(1H-pyrrol-1-yl)propanamide
4-(2-methoxyphenoxy)-1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)piperidine-4-carboxylic acid
N-({1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}methyl)-2,3-dimethoxybenzamide
8-[(3-fluorophenyl)methyl]-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(1H-indol-2-yl)ethyl]-1-(methoxymethyl)-N-methylcyclobutane-1-carboxamide
methyl 6-({[2-(diethylamino)pyridin-3-yl]methyl}amino)pyridine-3-carboxylate
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-(pyrimidin-2-yl)piperidine-4-carboxamide
2-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
N-cyclohexyl-3-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propanamide
1-[(8-fluoroquinolin-2-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1-{3-[3-(1-methyl-1H-pyrazol-4-yl)phenyl]-1H-pyrazol-1-yl}butan-2-ol
3-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)(pyridin-4-ylmethyl)amine
(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-3-(2-methylpropyl)piperidin-3-yl)methanol
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-4-carboxamide
1-(2,3-dimethylphenyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-4-amine
ethyl N-({1-[(3S,5S)-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}methyl)-N-methylcarbamate