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3-[2-(1,2-oxazolidin-2-yl)-2-oxoethyl]-4-[(3-phenoxyphenyl)methyl]piperazin-2-one
3-(4-fluorophenyl)-1-[(4-methanesulfonylphenyl)methyl]pyrrolidine
1-[(2,3-difluorophenyl)methyl]-4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2,6-dimethyl-N-(oxolan-2-ylmethyl)pyrimidine-4-carboxamide
(4aS,8aR)-6-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
3-{1-[(4-hydroxyphenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
3-[2-(thiophen-3-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]phenol
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-3-(3-methylpiperidin-1-yl)propan-1-one
7-methyl-3-{[4-(1-methylpiperidin-4-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
2-(3-chloro-2,6-difluorophenyl)-1-[(1-propyl-1H-pyrazol-4-yl)methyl]-1H-imidazole
4-hydroxy-3-methoxy-N-{1-[(4-methylphenyl)methyl]cyclopropyl}benzamide
2-{2-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
8-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(1-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}piperidin-4-yl)pyrrolidin-2-one
3-(2-chlorophenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]propanamide
(2R)-1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidine-2-carboxamide
N-[(3S,4R)-1-(naphthalene-1-sulfonyl)-4-propylpyrrolidin-3-yl]acetamide
(1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)methanamine
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
(2S,4R)-1-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-(dimethylamino)pyrrolidine-2-carboxylic acid
4-(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)-6-fluoro-1,2,3,4-tetrahydroquinolin-2-one
1-(1-{[3-(4-chlorophenoxy)phenyl]methyl}piperidin-4-yl)-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-{2-[1-(4-chloro-2-methoxybenzoyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
methyl 4-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]piperazine-1-carboxylate
N,1-dimethyl-2-oxo-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
5,7-dimethyl-N-[3-(propan-2-yloxy)propyl]pyrido[2,3-d]pyrimidin-4-amine
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-3-(methylsulfanyl)propanamide
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
3-(4-hydroxyphenyl)-N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2-phenylpropanamide
3-ethyl-8-(1-methoxypropan-2-yl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[(3-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
(3S,4S)-1-(5-cyanopyridin-2-yl)-4-cyclopropylpyrrolidine-3-carboxylic acid
5-chloro-N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2-methoxybenzene-1-sulfonamide
N-(1-phenylbutyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-ethyl-N-[(2-fluorophenyl)methyl]-N-methyl-1H-indole-2-carboxamide
2-{[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]methyl}-8-fluoroquinolin-4-ol
3-[3-({[1-(3-cyanopyridin-2-yl)piperidin-4-yl]amino}methyl)-1H-indol-1-yl]propanamide
8-(3-chloro-4-methylbenzoyl)-3-[2-(dimethylamino)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-[4-(thiophen-3-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
2-[3-(4-fluorophenoxymethyl)-5-(5-hydroxypyrazin-2-yl)-1H-1,2,4-triazol-1-yl]acetic acid
6-[4-(hydroxymethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-N,N-dimethylpyrazine-2-carboxamide
3-[N-(2-phenylethyl)-1-(3-propanamidophenyl)formamido]propanamide
1-{1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]piperidin-4-yl}-3-methylbutan-1-ol
8-(2,6-dimethylpyrimidine-4-carbonyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(1S,6R)-3-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3,9-diazabicyclo[4.2.1]nonane
2-(dimethylamino)-7-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-cyclopentyl-4-oxo-4-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}butanamide
1-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[2-(pyrrolidin-1-yl)ethyl]-1,4-diazepane-6-carboxylic acid
3-[2-(3,4-difluorophenyl)ethyl]-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidine