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{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[2-(1,3-thiazol-4-yl)ethyl]amine
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl][(4-fluoro-3-methoxyphenyl)methyl]methylamine
1-(carbamoylmethyl)-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
{[(3R,4S)-1-(3-fluoropyridin-4-yl)-4-propylpyrrolidin-3-yl]sulfamoyl}dimethylamine
3,5-dimethyl-4-(1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}pyrrolidin-2-yl)-1,2-oxazole
5-({3-[(3,4-difluorophenyl)amino]piperidin-1-yl}methyl)-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
2-(3-methylthiophen-2-yl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1H-imidazole
N-(1-{7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
4-[5-(thiomorpholine-4-carbonyl)pyrimidin-2-yl]morpholine
1-{4-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
N-cyclohexyl-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
3-methyl-5-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]-1H-pyrazole
N-(5-chloro-2-methoxyphenyl)-3-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-3-yl}propanamide
3,5-dimethyl-N-{3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}benzamide
N'1-[(3R,4S)-4-cyclopropyl-1-[(5-propylfuran-2-yl)methyl]pyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
3-{[(dimethylcarbamoyl)(phenyl)methyl]amino}-N-(2,3-dimethylphenyl)propanamide
9-{[2-(butan-2-yloxy)-3-methoxyphenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
4-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-(methylsulfanyl)-1,3-thiazole
4-{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazin-2-one
({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(oxolan-2-ylmethyl)propylamine
2,6-dimethyl-5-{2-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
2-phenoxy-N-[4-(4-{[3-(pyridin-3-yloxy)propyl]amino}piperidin-1-yl)phenyl]acetamide
1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}piperidine-3-carbonitrile
N-[(3R,4R)-3-hydroxy-1-(isoquinolin-1-yl)piperidin-4-yl]pyrazine-2-carboxamide
N3-methyl-N5-(2-methylpropyl)-N3-(naphthalen-1-ylmethyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(pyrrolidine-1-carbonyl)-1-(2,3,4-trimethoxybenzoyl)piperazine
3-[1-(cyclopropylmethyl)-1H-pyrazol-5-yl]-1-methyl-1-[(1-phenylpyrrolidin-3-yl)methyl]urea
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]ethane-1-sulfonamide
8-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(2,3-dimethoxyphenyl)methyl]-3-[2-(piperidin-1-ylmethyl)phenyl]urea
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]urea
[2-(7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]urea
N-{1-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-4-carboxamide
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pyrimidin-2-amine
2-[1-(carbamoylmethyl)-2-methyl-1H-indol-3-yl]-1H-1,3-benzodiazole-6-carboxylic acid
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(pyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
5-methyl-N-[(1R,2S)-2-phenylcyclopropyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-benzyl-5-(cyclopropylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine
3-{[(4-fluorophenyl)methyl]sulfanyl}-N-[(3R,4R)-4-hydroxypyrrolidin-3-yl]propanamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
2-{3-methyl-3,9-diazaspiro[5.6]dodecan-9-yl}-2-oxoacetamide
4-phenyl-N-{[1-(thian-4-yl)piperidin-3-yl]methyl}benzamide
5-{3-[(3-ethylphenyl)carbamoyl]propanoyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
7-(2-cyclohexylethyl)-2-(1-methylpiperidine-4-carbonyl)-2,7-diazaspiro[4.5]decane
2-[(1-acetylpiperidin-4-yl)oxy]-N-(2,3-dihydro-1H-inden-1-yl)-5-methoxybenzamide
5,6-dimethyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-[(1-methyl-1H-indol-3-yl)sulfanyl]ethan-1-one
2-[4-(2-hydroxy-4-methylbenzoyl)-5-methyl-2-oxopiperazin-1-yl]benzonitrile