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N-(2,2-dimethyloxan-4-yl)-N-ethyl-2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetamide
1-(furan-3-carbonyl)-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
(3aR,6aS)-5-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
N-cyclohexyl-3-[(6-methoxy-1-methyl-1H-indol-2-yl)formamido]propanamide
1-(4-{4-[2-cyclobutyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(oxan-4-ylmethyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
5-({4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}methyl)-1,2,4-oxadiazole-3-carboxamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[(1-phenylcyclopropyl)amino]methyl}piperidin-2-one
5-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}methyl)-N,N-dimethylpyridin-2-amine
3-(3-hydroxyquinoxalin-2-yl)-N-[1-(1H-indol-2-yl)ethyl]-N-methylpropanamide
1-(1-benzylpiperidin-4-yl)-N-[3-(methylsulfanyl)propyl]piperidine-3-carboxamide
2-{4-[(3-methyl-1H-pyrazol-5-yl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-{4-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperazin-1-yl}ethan-1-one
2,6-dimethoxy-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pyridine-3-carboxamide
1-{2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]acetyl}-4-phenylpiperidine-4-carbonitrile
3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-N-(trimethyl-1H-pyrazol-4-yl)benzamide
2-(cyclohex-1-en-1-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]acetamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}[(3-methyloxetan-3-yl)methyl]amine
3-(2-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindol-1-one
2-(6-methoxynaphthalen-2-yl)-4-(4-methylpyrimidin-2-yl)morpholine
1-{3,5-dimethyl-4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
N-{1-[2-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-1H-indol-3-yl]propan-2-yl}acetamide
N-(2H-1,3-benzodioxol-5-yl)-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-5-methyl-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
methyl 2-({[1-(cyclopropylmethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}amino)acetate
N-(furan-2-ylmethyl)-4-({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amino)pyridine-2-carboxamide
2-acetamido-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)acetamide
8-{[3-(2-hydroxyethoxy)phenyl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[(1-ethyl-1H-indol-5-yl)methyl](methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
3-[4-(6-ethylpyrimidin-4-yl)piperazine-1-carbonyl]piperidine-1-carboxamide
1-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
4-[(dimethylamino)methyl]-1-(5-propyl-1,2-oxazole-3-carbonyl)azepan-4-ol
4-methoxy-N-(2-{7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-4,6-dimethyl-1,2-dihydropyridin-2-one
1-(carbamoylmethyl)-N-[2-(4,5,6,7-tetrahydro-1-benzothiophen-3-yl)ethyl]piperidine-3-carboxamide
2-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]-N-[2-(4-methoxyphenyl)ethyl]acetamide
3-chloro-4-fluoro-N-[(4-hydroxyazepan-4-yl)methyl]-1-benzothiophene-2-carboxamide
3-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-6-ethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-[(3R,4S)-1-(2-ethylpyridine-4-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
4-{[(3R,5R)-3-(pyrrolidin-1-ylmethyl)-5-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}pyridine
2-(1H-imidazol-2-yl)-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)benzamide
N-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-6-oxo-1,6-dihydropyridine-2-carboxamide
N-[2-(2-chlorophenoxy)ethyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-(butan-2-yl)-3-(N-methylmethanesulfonamido)-N-(pyridin-3-ylmethyl)propanamide
methyl 4-[(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]benzoate
2-cyclopropyl-4-phenyl-9-(1,3-thiazol-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
9-(2-chloro-6-fluorobenzoyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(dimethylamino)ethyl]-N-ethyl-4-[(2-methylprop-2-en-1-yl)oxy]benzamide