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9-{[3-(methylsulfanyl)phenyl]methyl}-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}amine
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropylpyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl}-1H-1,3-benzodiazole-7-carboxamide
9-(4-chloro-2-methylbenzoyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-4-cyclobutyl-1-(2-hydroxyethyl)-3-methylpiperidin-4-ol
2-{[4-(6-methoxypyridin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-methyl-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-5-propyl-1,3,4-oxadiazole-2-carboxamide
1-[1-(2-methoxyethyl)-5-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-methyl-1,4-diazepane
N-(3-hydroxy-2,2-dimethylpropyl)-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(pyridin-2-ylmethyl)acetamide
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidine-1-carbonyl}cyclopropan-1-amine
(3S,4R)-1-cyclobutanecarbonyl-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
3-[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-(thiophen-2-ylmethyl)propanamide
(1S,2S,9S)-N-(4-cyano-2-ethylphenyl)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecane-11-carboxamide
5-(2-methylpropyl)-1'-(5-methylthiophene-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(4aR,7aS)-1-methyl-4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[2-(1H-imidazol-1-yl)ethyl]-1-[4-(trifluoromethyl)benzoyl]piperidine
(1S,5R)-N-(3-cyanophenyl)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]-1H-indazole
N-{[2-(dimethylamino)-7-fluoroquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-(3-methyl-1H-pyrazol-1-yl)acetamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-3-methyl-1H-pyrazole-4-carboxamide
1-{4-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]butyl}azepane
N-cyclopropyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-[(3-chlorophenyl)methyl]-3-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]propanamide
(5S)-5-[({[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(pyridin-2-ylmethyl)amino)methyl]pyrrolidin-2-one
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[4-(methylsulfanyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
3-methyl-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-1-propyl-1H-pyrazole-4-carboxamide
N-methyl-2-(oxolan-2-ylmethoxy)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
5-(1-benzofuran-2-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1,2,4-triazin-3-amine
2-[({1-[1-(4-fluorophenyl)cyclopropanecarbonyl]piperidin-4-yl}oxy)methyl]pyridine
[(3S,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(oxane-4-carbonyl)piperidin-3-yl]methanol
2-(adamantan-1-yl)-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
1-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-(2-hydroxyethyl)-3-[(5-methylthiophen-2-yl)methyl]urea
2-[3-(2-chlorophenyl)-1H-pyrazol-1-yl]-N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
4-{3-[4-(3-chlorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(2,2-dimethyloxan-4-yl)-2,3-dihydro-1H-isoindole-1,3-dione
N-methyl-N-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]thian-4-amine
5-butyl-1-(2-methoxyphenyl)-4-(oxane-4-carbonyl)piperazin-2-one
1-({[2-hydroxy-2-(naphthalen-2-yl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
(4aS,7aR)-1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-methoxyethyl)-9-oxo-N-(oxolan-2-ylmethyl)-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
2-[(1S,5R)-6-[2-(4-chlorophenoxy)ethyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]acetamide
N-[(5-methylthiophen-2-yl)methyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)-N-(pyridin-2-ylmethyl)acetamide
N-[1-(1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2H-1,3-benzodioxole-5-carboxamide
2-(cyclohex-1-en-1-yl)-1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}ethan-1-one
5-[(2,3-difluoro-6-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-2,4-dimethylpyrimidine-5-carboxamide