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N-[3-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-oxopropyl]methanesulfonamide
3-(aminomethyl)-4-(naphthalen-1-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(dimethylamino)propyl]-1-(3-fluorobenzenesulfonyl)-N-methylpiperidin-3-amine
6-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-2,3,4,9-tetrahydro-1H-carbazole
5-(4-fluorobenzoyl)-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
(3aR,6aS)-5-(3-cyanobenzoyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
2-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridine-3-carbonitrile
1-{[5-(3,3-dimethylbutyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3,3-dimethylurea
6-(2-methoxyphenyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(3-fluorophenyl)-1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]propan-1-one
6-cyclopentyl-2-methoxy-3-{[(2-methylpyrimidin-4-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[2-(furan-2-yl)pyrrolidin-1-yl]propan-1-one
5-{[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
4-(cyclopropylmethyl)-1-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-(3-methylpyridine-2-carbonyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-[5-(3-methylphenyl)-4H-1,2,4-triazol-3-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carboxamide
3-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-1-[1-(1-methyl-1H-pyrazol-4-yl)propyl]urea
1-(2,7-dimethylquinoline-4-carbonyl)-N-(3-hydroxypropyl)piperidine-3-carboxamide
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutanecarboxamide
2-{2-[(dimethylamino)methyl]phenyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[N-(2-phenylethyl)-1-5,6,7,8-tetrahydroquinolin-3-ylformamido]propanamide
2-{4-[(3-chloro-1-benzothiophen-2-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
N-[1-(2-fluorophenyl)piperidin-4-yl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
(2S,4R)-4-{[(3-fluorophenyl)methyl]amino}-N-methyl-1-(propan-2-yl)pyrrolidine-2-carboxamide
(3S,5R)-N3-[(1-ethylpyrrolidin-2-yl)methyl]-N5-(4-fluorophenyl)-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
4-[(4-fluorophenyl)methyl]-N-(5-methyl-1,3,4-thiadiazol-2-yl)-3-oxopiperazine-1-carboxamide
[(3-chloropyridin-4-yl)methyl][3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]methylamine
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
2-{[(1R,5S,6S)-6-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-3-azabicyclo[3.1.0]hexan-3-yl]methyl}phenol
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-2H-1,3-benzodioxole-5-carboxamide
N-[(4-fluorophenyl)methyl]-3-(1-phenylmethanesulfonylpiperidin-4-yl)propanamide
3-(1,3-benzothiazol-2-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
3-methyl-1-propyl-N-[1-(thian-4-yl)piperidin-4-yl]-1H-pyrazole-4-carboxamide
N-[(4-hydroxyazepan-4-yl)methyl]-3-(pyridin-3-yl)propanamide
1-(3-phenylbutyl)-4-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
2-(3-ethoxyphenyl)pyridin-4-amine
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methyl-N-(pyridin-3-ylmethyl)acetamide
3-(but-2-yn-1-yl)-5-[(3-fluorophenyl)methyl]-5-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
4-methyl-2-{2-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
N-{imidazo[1,2-a]pyrazin-3-ylmethyl}-2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)sulfanyl]propanamide
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methyl}-6-methylpyridine-3-carboxamide
2-(3-methoxypropyl)-9-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}pentan-1-one
N-(cyclopropylmethyl)-1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
(1R,2S)-1-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}-2,3-dihydro-1H-inden-2-ol
8-[5-(dimethyl-1,2-oxazol-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]quinoline
N-[(3S,4R)-1-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-{[5-(4-fluorophenyl)furan-2-yl]methyl}imidazo[1,2-a]pyridine-6-carboxamide