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3-(2-fluorophenyl)-N-methyl-N-[(3-methylpyridin-2-yl)methyl]-3-phenylpropanamide
N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl 2-{[4-(3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]sulfonyl}benzoate
4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(3-phenylpropyl)piperidine
1-[(4aS,8aS)-4a-hydroxy-7-(pyridin-4-ylmethyl)-decahydro-2,7-naphthyridin-2-yl]-2-methoxy-2-methylpropan-1-one
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
5-{[3-(1-methylpiperidin-3-yl)propanamido]methyl}thiophene-2-carboxylic acid
N-methyl-3-(5-methyl-1H-1,2,4-triazol-3-yl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}propanamide
2-({3-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}sulfanyl)-5-methyl-1,3,4-thiadiazole
N-(1-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
1-(diethylamino)-3-{5-[(4-fluoropiperidin-1-yl)methyl]-2-methoxyphenoxy}propan-2-ol
(3R,4S)-4-cyclopropyl-1-(2,6-difluoro-4-methoxybenzoyl)pyrrolidin-3-amine
2-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-cyclopropyl-1H-pyrazol-1-yl]-4-(5-methylfuran-2-yl)pyrimidine
N3-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-N5-[2-(4-phenylpiperidin-1-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
4-amino-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}butanamide
N-methyl-3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]propanamide
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-3,4,7-trimethyl-1H-indole-2-carboxamide
1-(4-{[(3-tert-butyl-1,2,4-oxadiazol-5-yl)methyl]amino}-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-(3-methylbutanoyl)-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-methylbut-2-en-1-one
N,6-dimethyl-N-[(3-methyloxetan-3-yl)methyl]-2-phenylpyrimidin-4-amine
(3R,4R)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-(2-methoxyethyl)-8-[(5-methylfuran-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-methoxy-5-methyl-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
1-[(2-fluorophenyl)methyl]-4-(quinoline-4-carbonyl)piperazin-2-one
3-(3-{[methyl({[3-(prop-2-en-1-yloxy)phenyl]methyl})amino]methyl}-1H-indol-1-yl)propanamide
4-{[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-5-phenyl-1,2-oxazole-3-carboxamide
2-methoxy-4-({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)pyridine-3-carbonitrile
(3R)-1-[3-(thiophen-3-yl)propyl]pyrrolidin-3-ol
N,6-dimethyl-2-oxo-N-[1-(pyridin-3-yl)pentyl]-1,2-dihydroquinoline-4-carboxamide
propan-2-yl 7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxylate
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-6-methoxy-N-methylpyrimidin-4-amine
N-(2-methoxyethyl)-5-phenyl-N-(1,3-thiazol-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
methyl 3-(cyclobutylmethoxy)-5-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]carbamoyl}benzoate
5-ethyl-1'-(7-fluoro-4-methylquinolin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(oxan-4-ylmethyl)amine
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)furan-3-carboxamide
1-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
methyl 3-(2,4-dimethylbenzamido)-6-{[methyl(oxolan-3-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
2-(1H-indol-3-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
7-cyclohexyl-2-(5-methylpyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N,N-dimethyl-5-({[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]amino}methyl)pyrimidin-2-amine
5-oxo-1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]pyrrolidine-3-carboxylic acid
1-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
N-[(6-chloropyridin-3-yl)methyl]-N-methyl-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-[(3,7-dimethyl-1H-indol-2-yl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide