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1-{2-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-2,3-dihydro-1H-inden-2-yl}piperidine
1'-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
6-(3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)pyridine-2-carbonitrile
1-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-3-(azocan-1-yl)propan-1-one
8-[(4-hydroxyphenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(pyridin-3-yl)-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
3-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-oxopiperidin-1-yl)ethyl]acetamide
2-ethyl-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}pyrimidine
1-{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
3-phenyl-N-(1-{1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
(1R,5R)-N,N-dimethyl-6-[2-(thiophene-2-sulfonamido)acetyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-(2-methoxyphenyl)-2-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]acetic acid
3-{[4-(3,4-diethoxyphenyl)-1H-imidazol-2-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
(3aS,6aS)-2-acetyl-5-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3S,4R)-1-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-4-propylpyrrolidin-3-yl]acetamide
9-[(2R)-2-amino-3-(furan-2-yl)propanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-{4-[(5-cyclopentylthiophen-2-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-7-fluoro-N,2-dimethylquinoline-4-carboxamide
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1H-imidazole-2-carboxamide
7-(1-benzothiophen-3-yl)-4-[2-(2-hydroxyethoxy)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3S,9aR)-3-[(benzyloxy)methyl]-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1,2-oxazole-3-carboxamide
4-[2,4-dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-3-methyl-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-6-one
2-methoxy-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]pyridine-3-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}acetamide
N-ethyl-N-(1-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-3-yl)acetamide
(1S,5R)-6-(cyclobutylmethyl)-3-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-4-[(4-fluorophenyl)sulfanyl]piperidine
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}bis(prop-2-en-1-yl)amine
2-(pyridin-2-yl)-5-({4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}methyl)pyrimidine
3-[3-({[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
4-ethyl-6-(4-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)pyrimidine
5-(3-fluorophenoxymethyl)-N-methyl-N-(pentan-3-yl)-1H-pyrazole-3-carboxamide
1-butyl-3-(2,6-dimethylpyridin-3-yl)-1-(pyridin-4-ylmethyl)urea
4-(1H-imidazol-2-yl)-1-(3-phenylbenzoyl)piperidine
1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-yl)piperazine
4-{[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}phenol
methyl({[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl})[1-(1,3-thiazol-2-yl)ethyl]amine
N-(2,4-dichlorophenyl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carboxamide
1-{[3,5-dichloro-4-(propan-2-yloxy)phenyl]methyl}-4-(hydroxymethyl)azepan-4-ol
(3S,4S)-3-hydroxy-4-[methyl(pyrazin-2-ylmethyl)amino]-N-(2-methylphenyl)pyrrolidine-1-carboxamide
N-{[5-(methylcarbamoyl)furan-2-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
2-[4-(methylsulfanyl)phenyl]-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
8-[(5-acetylthiophen-3-yl)methyl]-2-(pyridin-2-yl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]pyrimidine-5-carboxamide
(2S,4R)-4-amino-1-[(2-cyanophenyl)methyl]-N-ethylpyrrolidine-2-carboxamide
3-[({2-[(4-methoxyphenyl)sulfanyl]ethyl}amino)methyl]piperidin-3-ol
3-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-N-[(4-chlorophenyl)methyl]propanamide