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ethyl 2-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]amino}acetate
3-cyclopropyl-4-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-pyrazole
N-[(3R,4R)-3-hydroxy-1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl]pyrazine-2-carboxamide
3-(azepane-1-carbonyl)-N-[(2-methoxyphenyl)methyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-sulfonyl}benzonitrile
3-{[3-(3-methylpyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-(propan-2-yl)piperazin-2-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
5-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
1-(furan-2-carbonyl)-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}piperazine
5-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}-2-methoxybenzoic acid
3-{[(3-hydroxy-3-methylbutyl)(methyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
3-(4-{2-[(prop-2-en-1-yl)amino]benzoyl}piperazin-1-yl)pyrazine-2-carbonitrile
3-(3-methylphenyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
ethyl 2-[4-({methyl[(3-methylpyridin-4-yl)methyl]carbamoyl}amino)phenyl]acetate
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-cyclopropyl-N-[(4-methoxypyridin-2-yl)methyl]pyrimidin-4-amine
1-[2-hydroxy-3-(2-methoxy-4-{[(prop-2-en-1-yl)amino]methyl}phenoxy)propyl]piperidin-4-ol
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-cyclopropyl-5-[4-(trifluoromethyl)pyrimidin-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-amine
2-amino-N-cyclopropyl-3-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-(5-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
4-ethoxy-3-(pyridin-4-yl)benzoic acid
1-[(2-chloro-4-fluorophenyl)methyl]-N-methyl-N-(quinolin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(2-{[3-(2-fluorophenyl)-1H-pyrazol-4-yl]formamido}ethyl)-2-methylpropanamide
N-{[5-chloro-7-(1H-indol-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
6-[2-(4-methylpentyl)morpholine-4-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
1-(3-oxo-3-{2-[2-(pyridin-2-yl)ethyl]piperidin-1-yl}propyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-benzyl-8-(2,2-dimethylpropyl)-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
5-(2-methoxypyridin-3-yl)pyridine-3-carboxylic acid
N-methyl-N-{1-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-2-(1H-pyrazol-1-yl)acetamide
1-[4-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)thiophen-2-yl]ethan-1-one
N3-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]piperidine-1,3-dicarboxamide
(1R,5S)-N-[5-(cyclopropylcarbamoyl)-2-methoxyphenyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[(2-methoxyphenyl)methyl]-4-[3-(pyridin-4-yl)azetidine-1-carbonyl]pyrrolidin-2-one
5-fluoro-2-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
4-(4-methoxy-2-methylphenyl)-3-(pyrazin-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-{8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}pyridine-3-carbonitrile
7-(2,8-dimethylquinoline-4-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-oxo-2-phenylacetamide
1-(2-methylpyridin-4-yl)-4-(pyridin-4-ylmethyl)piperazine
N-[(2R)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-1-oxobutan-2-yl]acetamide
2-(4-ethenylbenzoyl)-2,7-diazaspiro[4.5]decane
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-(4-methoxyphenyl)-N-methylacetamide
6-{2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carboxylic acid
4-{[2-(dimethyl-1,3-thiazol-5-yl)phenyl]methyl}morpholine