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N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-3-yl}propanamide
3-(3-fluorophenyl)-1-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}propan-1-one
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-[(4-fluorophenyl)methyl]-4-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-(propan-2-yl)-1,4-diazepane
3-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-[5-methoxy-2-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
6-ethyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-(furan-2-ylmethyl)-5-{3-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
1-cyclobutanecarbonyl-N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)piperidine-4-carboxamide
(4aR,7aS)-1-(2-methylpropanoyl)-4-(1,2-oxazole-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[3-(1H-imidazol-1-yl)propyl]-9-(3,3,3-trifluoropropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(1H-imidazol-2-yl)ethyl]-2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carboxamide
3-(3,5-dimethylphenyl)-N-[(1-methylpiperidin-3-yl)methyl]propanamide
1-[4-({[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amino}methyl)thiophen-2-yl]ethan-1-one
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]naphthalene-1-sulfonamide
methyl 6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]-N-(2-methylprop-2-en-1-yl)acetamide
1-[(2-chloro-4-fluorophenyl)methyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
6-methoxy-4-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
3-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
(1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(4-methoxyphenyl)methyl]piperidin-4-yl)methanol
4-(4-phenylbenzenesulfonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
11-[(9H-fluoren-9-yl)amino]-4-(pyridin-4-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3,5-dimethyl-1-(prop-2-en-1-yl)-1H-pyrazole
methyl({[6-methyl-4-(thiomorpholin-4-yl)quinazolin-2-yl]methyl})[(5-phenyl-1,2-oxazol-3-yl)methyl]amine
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)naphthalene-1-carboxamide
3-[({1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-(pyridazine-3-carbonyl)-1,4-diazepan-5-one
(3R,4S)-4-{[(3,4-difluorophenyl)methyl](ethyl)amino}oxolan-3-ol
1-[benzyl(methyl)amino]-3-(5-{[ethyl(methyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
4-methyl-5-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-2-(propan-2-yl)-1,3-thiazole
N-(2,5-dimethylphenyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carboxamide
2-(3-chloro-5-fluoro-4-methoxyphenyl)-1H-imidazole
8-{[4-(4-chlorophenyl)phenyl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(4-methylphenoxy)piperidine
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}azetidin-3-amine
5-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
2-(2-hydroxyethyl)-9-(3-methoxy-4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-(quinolin-2-ylmethyl)pyrrolidin-3-yl]urea
N-cyclopropyl-3,5-difluoro-4-methoxy-N-[(2-methoxyphenyl)methyl]benzamide
N,1-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H-pyrrole-2-carboxamide
5-methyl-5-[1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-4-yl]imidazolidine-2,4-dione
3-benzyl-1-(3-methoxypropyl)-8-(quinoxalin-6-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-7-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 3-({5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}amino)propanoate
2-{[6-(4-fluorophenyl)-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}-N-methylacetamide
1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-3-(methylsulfanyl)propan-1-one