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4-(1-aminocyclobutanecarbonyl)-7-(1,3-benzothiazol-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
4-(4-ethoxy-3-methylphenyl)-N-(1H-imidazol-2-ylmethyl)butanamide
1-[2-({5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}amino)ethyl]pyrrolidine-2,5-dione
2-[(4-{[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]-1,2,3,4-tetrahydroisoquinoline
N-(2-methanesulfonamidoethyl)-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
5-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-2-methyl-1H-1,3-benzodiazole
N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-5-phenyl-1,2-oxazole-3-carboxamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl][(4,5-dimethylfuran-2-yl)methyl]methylamine
2-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-N,N-dimethylaniline
[(2S)-1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
N-[(2,4-difluorophenyl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
6-[2-(aminomethyl)-4-fluorophenyl]quinazolin-4-amine
2-amino-3-ethyl-N-[(2-propyl-1,3-thiazol-4-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-(2-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)methanesulfonamide
2-(4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
N-[(5-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
N-[2-(dimethylsulfamoyl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-{[4-(1H-1,3-benzodiazol-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-4-methylphenol
3-phenyl-1-[1-(1H-pyrazole-3-carbonyl)piperidin-3-yl]propan-1-one
3-benzyl-4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}piperazin-2-one
2-(4-methylphenyl)-N-[3-(1H-1,2,4-triazol-1-yl)propyl]quinoline-4-carboxamide
N,N-dipropyl-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
(3ar,6ar)-N-[(4-phenylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-(5-methylhexan-2-yl)-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
(1R,5R)-6-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
6-oxo-N-(pentan-3-yl)-N-(2-phenylethyl)-1,6-dihydropyridine-2-carboxamide
5-[4-(3,4-dichlorophenyl)piperazine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
(4aR,7aS)-4-{[2-(2-hydroxyethoxy)phenyl]methyl}-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)-1H-1,3-benzodiazole-6-carboxylic acid
2-(1,2-oxazole-3-carbonyl)-N-(1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]-2-(propan-2-yloxy)propan-1-one
2-(dimethyl-1,3-thiazol-5-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}acetamide
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-fluorophenyl)urea
1-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{4-[(2-chloro-6-fluorophenyl)methyl]-1,4-oxazepan-6-yl}methanol
(3S,9aR)-3-(4-aminobutyl)-8-benzyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-cyclopentyl-4-({methyl[(2-methyl-1H-imidazol-4-yl)methyl]amino}methyl)pyrrolidin-2-one
1-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidin-1-yl)-3-(methylsulfanyl)propan-1-one
4-(1H-pyrazol-1-yl)-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
5-{3-[4-(2-chlorophenoxy)piperidin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(2-methylphenyl)methyl]benzamide
1-[(3-methoxyphenyl)methyl]-5-({spiro[indene-1,4'-piperidine]-1'-yl}carbonyl)piperidin-2-one
2-fluoro-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)benzamide
2-methoxy-4-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridine
5-[(dimethylamino)methyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
3-{1-[2-(methylamino)acetyl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
3-(3-tert-butyl-1-methyl-1H-pyrazol-5-yl)-1-methyl-1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}urea
N-(1-benzothiophen-5-ylmethyl)-1-cyclopropanecarbonylpiperidine-4-carboxamide