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3-(oxolan-3-yl)-5-[3-(propan-2-yloxy)phenyl]-1,2,4-oxadiazole
N-(furan-2-ylmethyl)-6-methyl-N-(3-methylbutan-2-yl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
ethyl 1-(2-methyl-1H-1,3-benzodiazole-6-carbonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
2-(1H-imidazol-1-yl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
5-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-8-(2-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-3-(1-methyl-1H-imidazol-2-yl)piperidine
(cyclopropylmethyl)({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amine
N-[2-(4-chlorophenyl)ethyl]-N-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)methylamine
N-cyclopentyl-2-[methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl})amino]propanamide
(3R,4R)-1-(3-methoxy-5-methylthiophene-2-carbonyl)-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
3-{5-[(2,3-difluoro-6-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
4-[2-(3,4-difluorophenyl)pyridine-4-carbonyl]morpholine
2-{[(3,3-diphenylpropyl)amino]methyl}-4-(6-methoxypyridin-2-yl)phenol
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-5-(4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
ethyl 2-{2-[(1-methylpiperidin-2-yl)formamido]ethyl}-1,3-thiazole-4-carboxylate
N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
1-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]-4-methyl-1,4-diazepane
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)pyrrolidin-3-amine
8-(2,3-dihydroxypropyl)-3-[2-(4-ethylpiperazin-1-yl)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-fluorophenyl)-4-{[3-({1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-3-yl}methoxy)phenyl]methyl}piperazine
N-[(3-propyl-1,2-oxazol-5-yl)methyl]-6-(4-propyl-1,4-diazepan-1-yl)pyridine-3-carboxamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
8-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(3-methyl-1H-pyrazole-5-carbonyl)-3-phenylpiperidine
2-[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
8-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-benzyl-3-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-3-phenylprop-2-yn-1-one
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(thiophen-3-yl)propanamide
2-{1-benzyl-5-[3-(2-oxoimidazolidin-1-yl)phenyl]-1H-1,2,4-triazol-3-yl}acetamide
N-[1-(benzenesulfonyl)piperidin-4-yl]-1H-1,2,3-triazole-5-carboxamide
(3aR,6aR)-2-methanesulfonyl-5-{[3-(methylsulfanyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-amine
3-methyl-4-{2-[3-(3-methylphenoxy)azetidin-1-yl]-2-oxoethyl}-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(furan-2-carbonyl)-4-(5-methyl-1,3-oxazole-4-carbonyl)piperazine
N,N-dimethyl-2-{[(5-propylthiophen-3-yl)formamido]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-(6-chloro-2-methylpyridin-3-yl)-3-methyl-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
methyl 3-(furan-3-amido)-6-{[methyl(oxolan-3-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
(1R,7S)-6-(5-oxo-1,4-diazepane-1-carbonyl)-3-[4-(propan-2-yl)phenyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-(methylamino)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyridine-4-carboxamide
2-methyl-6-(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-3-yl)pyrimidin-4-ol
4-[1-(3-oxo-3,4-dihydroquinoxaline-2-carbonyl)piperidin-3-yl]benzoic acid
1-[2-methoxy-5-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3,4,7-trimethyl-2-(2-phenylazetidine-1-carbonyl)-1H-indole