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7-(1-benzyl-1H-pyrazole-4-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
[(3S,7S)-5-(5-propyl-1,3,4-thiadiazol-2-yl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-3-yl]methanol
4-methoxy-N,3-dimethyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
N-cyclopentyl-N'-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]butanediamide
(1R,5R)-6-benzyl-3-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
1-(2-methoxyethyl)-3-methyl-8-{[3-(2-methylphenyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-5,6-dimethylpyrimidin-4-amine
3-{[4-(4-ethylpiperazin-1-yl)piperidin-1-yl]methyl}-6-methyl-1-(prop-2-en-1-yl)-1,2-dihydroquinolin-2-one
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-2-methylpyrimidine-5-carboxamide
1-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
1-(2,1,3-benzoxadiazol-5-ylmethyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
N-[(3S,4R)-1-[2-(4-hydroxyphenyl)acetyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
3-({4-[(4-methoxy-4-methylpentan-2-yl)amino]piperidin-1-yl}methyl)phenol
6-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-5,6,7,8-tetrahydro-1,6-naphthyridine
N-(1-benzyl-1H-pyrazol-3-yl)-2-{4-[4-(hydroxymethyl)phenyl]-1H-pyrazol-1-yl}acetamide
N-({2-[(2-methoxyphenyl)methyl]-6-oxo-1,6-dihydropyrimidin-4-yl}methyl)-5-methylpyridine-3-carboxamide
(3S)-3-[4-(5-tert-butyl-1H-pyrazol-3-yl)-1H-1,2,3-triazol-1-yl]azepan-2-one
4-{[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]methyl}benzonitrile
2-(4-tert-butylphenoxymethyl)-4-hydroxy-N-(oxolan-2-ylmethyl)pyrimidine-5-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(4-{[methyl(pyridin-3-ylmethyl)amino]methyl}-1H-pyrazol-1-yl)propanoic acid
1-(carbamoylmethyl)-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-3-carboxamide
4-ethyl-5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,2,3-thiadiazole
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
1-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]urea
1-{4-[4-(3-hydroxyphenyl)piperidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
2-[4-chloro-2-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]acetic acid
{1-[2-(2,3-dimethylphenoxy)ethyl]piperidin-2-yl}methanol
[(2-chloro-4,5-dimethoxyphenyl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
2,6-dimethoxy-4-{[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}phenol
[(2E)-3-(furan-2-yl)prop-2-en-1-yl](methyl){[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
9-methoxy-3-[2-(2-methoxyphenyl)acetyl]-N-methyl-7-oxo-N-(1,3-thiazol-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidin-4-yl)-2-phenylethan-1-ol
1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-amine
3-{1-[(3-phenoxyphenyl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1H-1,2,3-benzotriazole-5-carboxamide
N-({7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
N-[4-(1H-pyrazol-1-yl)butan-2-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,3-oxazole-4-carboxamide
N-{[1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methyl}-6-methylquinoline-4-carboxamide
methyl(oxan-2-ylmethyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
3-{[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]amino}-N-(2-methylphenyl)propanamide
2-oxo-1-phenyl-N-{[3-(trifluoromethoxy)phenyl]methyl}pyrrolidine-3-carboxamide
1-(2-{[6-(2-methoxyphenyl)pyridazin-3-yl]amino}ethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-(2-methoxyphenyl)-4-[1-(pyridin-4-ylmethyl)piperidin-3-yl]piperazine
N,N,4,5-tetramethyl-6-[4-(piperidin-1-yl)piperidin-1-yl]pyrimidin-2-amine
3-(1H-imidazol-1-yl)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]butan-1-one
(1S,5R)-6-(dimethyl-1,3-thiazole-5-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{1-cyclohexyl-4-[(1-ethyl-1H-imidazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[(3-methoxyphenyl)methyl]amine
[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine