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(1R,5S,6R)-3-({2-[(2-methylphenyl)methoxy]phenyl}methyl)-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
3-benzyl-1-methyl-8-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 4-({3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}methyl)benzoate
2-(furan-2-yl)-5-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}pyrimidine
6-{1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
1-{4-[(cycloheptylamino)methyl]-2-methoxyphenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
2-[4-(2,1,3-benzothiadiazol-4-yl)-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl]acetic acid
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
methyl (2S,4R)-4-[4,5-dimethyl-2-(1H-pyrrol-1-yl)thiophene-3-amido]-1-methylpyrrolidine-2-carboxylate
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2,3-dihydro-1-benzofuran-5-carboxamide
(2E)-N-cyclopropyl-N-({3-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-3-(thiophen-2-yl)prop-2-enamide
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
4-[(2,4-dimethoxy-3-methylphenyl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(4-methyl-1H-pyrazol-1-yl)-1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]piperidine-4-carboxylic acid
N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-3-methylthiophene-2-carboxamide
N-[(1R,3S)-3-[(5-methoxy-2-methylphenyl)carbamoyl]cyclopentyl]thiophene-3-carboxamide
N-(2,6-dimethoxypyridin-3-yl)-4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carboxamide
6-(2-chlorophenyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
[(2-butyl-1H-imidazol-4-yl)methyl](2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
3-fluoro-N-{1-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-oxo-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N,N-dimethyl-5-[(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)methyl]pyridin-2-amine
(2S)-2-{[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazol-3-yl]formamido}propanamide
3-[(2,4-difluorophenyl)methyl]-1-(9H-purin-6-yl)piperidine-3-carboxylic acid
3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-{2-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
2-(cyclohex-1-en-1-yl)-N-{[5-fluoro-7-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
2,6-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]quinoline-4-carboxamide
2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}acetamide
7-(5-methylthiophen-2-yl)-4-(piperidin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-cyclopentyl-N3,N3-diethyl-N5-[(3-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-cyclopropyl-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-4-(trifluoromethyl)benzamide
ethyl 5-(1H-indole-2-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}-4-(2-methylpropyl)piperazin-2-one
3-({[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-(1-methyl-1H-pyrazol-4-yl)propanamide
5-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-1,7-dimethyl-1H,2H,3H,4H-pyrido[2,3-d]pyrimidine-2,4-dione
1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-(pyridin-2-yl)propan-1-one
(3S,4R)-1-(1,3-benzoxazol-2-yl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
N-[(2-methoxyphenyl)methyl]-N-propyl-2,5-dihydro-1H-pyrrole-2-carboxamide
2-(5-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}furan-2-yl)benzonitrile
(1S,5R)-6-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
2-[(dimethylcarbamoyl)amino]-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)acetamide
5-(furan-2-yl)-3-({2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)-1,2-oxazole
N-{[3-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-1,3-thiazole-5-carboxamide
2-(ethylamino)-N-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}pyrimidine-5-carboxamide
1-[cyclohexyl(methyl)amino]-3-[2-methoxy-4-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
methyl (2S)-2-[methyl({6-oxo-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-7-yl}methyl)amino]propanoate
(2E)-1-[(4aR,8aS)-6-(oxane-4-carbonyl)-decahydro-1,6-naphthyridin-1-yl]-3-(2-fluorophenyl)prop-2-en-1-one
4-methyl-5-{9-methyl-3,9-diazaspiro[5.6]dodecane-3-carbonyl}pyrimidin-2-amine
3-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea