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(3R,5S)-N-(2-hydroxyethyl)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
(3R,4R)-4-amino-1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}piperidin-3-ol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-(naphthalen-2-yloxy)propanamide
(2R,3R)-3-(dimethylamino)-1'-[2-(methylamino)pyridine-3-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(1-{[1-(2-phenylbenzoyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
N-benzyl-2-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]acetamide
8-(2-methylpyridin-4-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
methyl 3-[(3S,4R)-1-[(2-hydroxyphenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
2-(pyridin-2-yl)-N-(pyridin-2-ylmethyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-[1-(3-cyclohexylpropanoyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)imidazolidine-2,4-dione
1-[2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carbonyl]piperidin-3-ol
5-(2,3-dihydro-1H-inden-2-yl)-3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(2,5-dimethylphenyl)methyl]piperidine-3-carboxamide
3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperidine
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
4-(methoxymethyl)-6-[2-(propan-2-yloxy)phenyl]pyrimidine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-ethyl-N-methyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N,N,4-triethyl-5-methylthiophene-3-carboxamide
[(2-methoxyphenyl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})(pyridin-3-ylmethyl)amine
(1S,5R)-1,3,3-trimethyl-6-(1-methyl-1H-imidazole-2-carbonyl)-6-azabicyclo[3.2.1]octane
9-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-benzyl-N-ethyl-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
methyl({3-[4-(8-methylquinolin-5-yl)-1H-1,2,3-triazol-1-yl]propyl})amine
8-acetyl-2-[(5-carboxyfuran-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
N-[5-(2-hydroxy-2-phenylpropanamido)-2-methoxyphenyl]furan-2-carboxamide
2-methyl-5-{[2-(1-phenylethyl)-1H-imidazol-1-yl]methyl}pyrazine
N-methyl-5-[2-(methylsulfanyl)phenoxymethyl]-N-(pyrazin-2-ylmethyl)-1,2-oxazole-3-carboxamide
(3S,4R)-N,N-dimethyl-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-amine
3-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propanamide
3-(2-methyl-1H-indol-1-yl)-1-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
2-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-2-yl)pyridine
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
1-{[1-(5-carbamoylpyridin-2-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxylic acid
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propylacetamide
5-acetyl-N-[2-(ethylsulfanyl)ethyl]thiophene-3-carboxamide
3-chloro-4-fluoro-N-(2-oxopyrrolidin-3-yl)-1-benzothiophene-2-carboxamide
N-({1-[3-(4-hydroxyphenyl)-2-phenylpropanoyl]piperidin-4-yl}methyl)acetamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-2-(piperidin-1-yl)pyridine
7-methyl-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
(1S,6R)-3-(6-chloropyridazin-3-yl)-3,9-diazabicyclo[4.2.1]nonane
4-{2-chloro-4-[(2-methoxyethyl)carbamoyl]phenoxy}-N,N-dimethylpiperidine-1-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(3,5-dimethylphenyl)methyl]-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
1-(1,4-dithiepan-6-yl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
3-({1-[2-(2-methyl-1H-indol-3-yl)acetyl]pyrrolidin-3-yl}methyl)benzamide
5-(2H-1,3-benzodioxol-4-ylmethyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide