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N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-2-(3-phenylpiperidin-1-yl)acetamide
1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-3-(1-methylcyclopropyl)propan-1-one
1-ethyl-N-[3-(2-methoxyphenyl)propyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
ethyl 3-[(3-methoxyphenyl)methyl]-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine-3-carboxylate
N-(cyclohex-1-en-1-ylmethyl)-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
7-[3-(5-methyl-1,2,4-oxadiazol-3-yl)benzenesulfonyl]-2,7-diazaspiro[4.5]decane
3-{2-[(dimethylamino)methyl]phenyl}-5-(morpholine-4-sulfonyl)benzoic acid
4-(1-{4-[6-(pyrrolidin-1-yl)pyridazin-3-yl]phenyl}ethyl)morpholine
2-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-4-methylphenol
(3R,4R)-4-(azepan-1-yl)-1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-ol
1-ethyl-8-[(3-methoxyphenyl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-(piperidine-1-carbonyl)pyridine
2-[3-(methylsulfanyl)phenyl]-1-[4-(piperidine-1-carbonyl)piperidin-1-yl]ethan-1-one
(1-{1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)(phenyl)methanol
4-(1-{1-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
3-[1-ethyl-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]propanamide
3-(carbamoylmethoxy)-N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]benzamide
5-{2-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{4-[4-(pyridin-2-yl)piperazine-1-carbonyl]piperidin-1-yl}-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-chloro-N-(1-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
N-(3-methoxypropyl)-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(2,2-dimethyloxan-4-yl)-6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
ethyl 1-(cyclopropylmethyl)-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
6-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)pyridine-2-carboxylic acid
5,7-dimethyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]-4-(pyrrolidine-1-carbonyl)quinoline
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[3-(methylsulfanyl)butyl]piperazine
N-(1-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-1H-indol-3-yl}propan-2-yl)acetamide
2-[1-benzyl-5-(2,6-difluoro-3-methoxyphenyl)-1H-1,2,4-triazol-3-yl]acetamide
1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
N-[(2-{3-[2-(4-methoxyphenyl)acetamido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-3-(pyridin-2-yl)propanamide
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-(quinoxalin-5-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[2-(dimethylamino)ethyl]-1-{7-methoxy-3-[({[2-(trifluoromethyl)phenyl]methyl}amino)methyl]quinolin-2-yl}-1,4-diazepan-5-one
1-cyclopentyl-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
N-[(2-methoxyphenyl)methyl]-4-[(3-methoxypropyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
4-{5-fluoro-2-[4-fluoro-2-(trifluoromethyl)phenyl]pyrimidin-4-yl}morpholine
N-methyl-3-[(pyrrolidin-3-yl)sulfamoyl]-N-(thian-4-yl)benzamide
N-[(3R,4R)-1-[(4-ethoxyphenyl)methyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
[(3R,5R)-1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-3-yl]methanol
4-{[4-(1-hydroxy-3-phenylpropyl)piperidin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl][2-methyl-2-(morpholin-4-yl)propyl]amine
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(4-{[(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amino]methyl}phenyl)acetamide
(3aR,6aR)-2-(4-chloro-3-fluorobenzoyl)-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-(2-hydroxypyridine-3-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-3-azaspiro[5.5]undecan-9-amine
4-methyl-2-(4-methylpiperazin-1-yl)-5-[3-(pyridin-2-yl)azetidine-1-carbonyl]pyrimidine
ethyl 5-(1H-1,3-benzodiazol-2-ylmethyl)-1-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-(1H-imidazol-1-yl)ethan-1-one
2-{[4-(2-methoxyphenyl)-5-(oxan-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid