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6-methyl-2-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}quinolin-4-ol
1-(2-methyl-4-{[2-(1H-pyrrol-1-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)ethan-1-one
2-(benzylamino)-1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]ethan-1-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(methylsulfanyl)propanamide
1-(5-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}thiophen-2-yl)ethan-1-one
3-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanamide
4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}-N-(4-methylphenyl)piperidine-1-carboxamide
N,5,6-trimethyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-{2-[3-(thiophen-2-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-4-carboxamide
1-(pyridin-4-ylmethyl)-4-[4-(1,3-thiazol-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
1-(5-chloropyridin-2-yl)-4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazine
2-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
N-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-amino-2-methyl-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
N4-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-5-butyl-6-methylpyrimidine-2,4-diamine
4-(5-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}pyrimidin-2-yl)morpholine
4-[2-(thiophen-2-yl)acetyl]morpholine-2-carboxylic acid
2-methyl-8-[1-(4-phenylphenyl)-1H-1,2,3,4-tetrazol-5-yl]-2,8-diazaspiro[4.5]decan-3-one
2-cyclohexyl-6-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]-1,3-benzoxazole
6-methyl-N-[(2-methylpyridin-4-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
1-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(2,6-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
4-[(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methyl]morpholine
[(3aS,6aS)-2-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
N-[(2-ethoxypyridin-3-yl)methyl]-5-methanesulfonyl-2-methylpyrimidin-4-amine
(1S,5R)-6-[2-(1H-imidazol-2-yl)benzoyl]-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
4-(4-ethoxy-3-methylphenyl)-N-[2-(3-hydroxypiperidin-1-yl)ethyl]butanamide
2-cyclopropyl-5-[4-(4-methylphenoxy)piperidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
(3R,4S)-3,4-dimethyl-1-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]piperidin-4-ol
{1-[(1-methanesulfonylpiperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}(phenyl)methanol
2-cyclopropyl-N-(2-ethoxyethyl)-6-oxo-1,6-dihydropyrimidine-5-carboxamide
3-{[4-(4-benzyl-5-{[(4-fluorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}pyridine
8-[(6-chloro-2H-chromen-3-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-methyl-4-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]piperazine
2-(1-cyclopentyl-4-ethylpiperazin-2-yl)ethan-1-ol
N-[2-(dimethylamino)ethyl]-N-methyl-1-(3-phenylpropyl)piperidin-3-amine
methyl 3-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-cyclopentyl-9-[3-(5-methylfuran-2-yl)butyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(5-methylpyrazin-2-yl)methyl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-amine
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)propan-1-one
(3R,4R)-4-methyl-3-(propan-2-yl)-1-(1,3-thiazol-2-yl)pyrrolidin-3-ol
2-[4-(hydroxymethyl)phenyl]-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
methyl 3-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propanoate
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
2-[(2R)-2-aminopropanoyl]-N-(cyclopropylmethyl)-N-propyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-ethoxypropanamide