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5-{1-oxa-7-azaspiro[3.5]nonan-7-yl}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
5-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}-5-(pyridin-3-yl)imidazolidine-2,4-dione
2-(3,4-dimethoxyphenyl)-N,6-dimethylpyrimidin-4-amine
2-methyl-4-{5-[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]furan-2-yl}but-3-yn-2-ol
N-[4-(furan-2-yl)phenyl]-1-[3-(pyrazin-2-yl)propanoyl]piperidine-3-carboxamide
(4aR,7aS)-1-{2-[(1R,5S,8S)-8-hydroxy-3-azabicyclo[3.2.1]octan-3-yl]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N,3,5-trimethyl-4-oxo-N-{[3-(prop-2-en-1-yloxy)phenyl]methyl}-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
N2,N2-dimethyl-N4-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
(2E)-1-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(pyridin-4-yl)prop-2-en-1-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-5-propyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
{1-[({[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]cyclopropyl}methanol
2-{[(1S,4S)-5-methyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]methyl}-N-(thiophen-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-N-(1-benzylpyrrolidin-3-yl)propanamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-(2-phenylethyl)-N5-(thiophen-2-ylmethyl)piperidine-3,5-dicarboxamide
5-ethyl-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]thiophene-3-carboxamide
(3S,4S)-4-(naphthalen-2-yl)-1-(pyridin-4-ylmethyl)piperidin-3-ol
2-fluoro-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-5-sulfamoylbenzamide
1-(3-methylbutyl)-8-(propan-2-yl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-phenylpropanamide
2-[2-(2-methoxyethyl)pyrimidin-5-yl]-N,N-dimethylquinoline-4-carboxamide
4-cyclopentyl-2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
4-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-N-(oxan-4-yl)morpholine-2-carboxamide
1-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}-2-(methoxymethyl)piperidine
[(dimethyl-1,3-thiazol-5-yl)methyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
(1S,5R)-N-(furan-2-ylmethyl)-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[(4-{furo[3,2-c]pyridin-4-yl}piperazin-1-yl)methyl]-4,5,6,7-tetrahydro-1,3-benzothiazole
2-[(4-{4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]phenoxy}piperidin-1-yl)methyl]pyridine
4-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-4-oxobutane-1-sulfonamide
2-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)pyridine-4-carbonitrile
2-benzyl-5-cyclopentanecarbonyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine
N-[2-(dimethylamino)ethyl]-5-(1-{[2-(methylamino)pyridin-3-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-cyclohexyl-N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazole-4-carboxamide
(2S)-2-[2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamido]propanamide
(isoquinolin-5-ylmethyl)(methyl){[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2,8-dimethylquinoline-4-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-[3-(2-methoxyphenyl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-[2-(3-fluorophenyl)ethyl]-1-(propan-2-yl)pyrrolidine-2-carboxamide
1-methyl-4-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-methyl-2-(1-oxo-1,2-dihydroisoquinolin-2-yl)-N-[3-(oxolan-2-yl)propyl]acetamide
1-cyclopentyl-5-[3-(3-ethylphenoxy)azetidine-1-carbonyl]piperidin-2-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}propanamide
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-ethyl-4-{[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}pyrrolidine-2-carboxamide
2-[(E)-2-[4-(2-cyclopropyl-1H-imidazol-1-yl)phenyl]ethenyl]pyridine
8-[2-(2,6-dimethoxyphenoxy)ethyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1R,3S)-3-methoxy-7-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-7-azaspiro[3.5]nonan-1-ol
N-(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
N-benzyl-N-(cyclobutylmethyl)-2-methanesulfonylacetamide
dimethyl(2-{4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]morpholin-2-yl}ethyl)amine
3-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
2-[4-fluoro-3-(hydroxymethyl)phenyl]-2-{methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}acetic acid