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2-(2,3-dihydro-1H-inden-1-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}acetamide
benzyl 3-{[(5-methyl-1,2-oxazol-3-yl)formamido]methyl}piperidine-1-carboxylate
4-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-amido]-N-cyclohexylpiperidine-1-carboxamide
1-ethyl-4-{[methyl({5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl})amino]methyl}pyrrolidin-2-one
2-{4-[(3,5-dichloropyridin-4-yl)methyl]piperazin-1-yl}-N-ethylacetamide
(2S,4R)-1-benzyl-N-methyl-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N6-cyclopentyl-N5-(oxolan-2-ylmethyl)-N5-(pyridin-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-cyclopropyl-4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
N-[4-(3-methoxyphenyl)phenyl]-1-[(6-methylpyridin-2-yl)methyl]piperidine-3-carboxamide
4-(2H-1,3-benzodioxol-5-yl)-2-methyl-6-(propan-2-yl)pyrimidine
2-amino-4-(3-cyclohexyl-1H-pyrazol-4-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N,4-dimethyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-(2-oxoimidazolidin-1-yl)benzamide
3,5-difluoro-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyridine-2-carboxamide
4-{5-[2-chloro-4-(4H-1,2,4-triazol-4-yl)phenyl]-3-cyclopropyl-1H-1,2,4-triazol-1-yl}-2-methylpyridine
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-3-(thiophen-3-yl)propanamide
N-[(4-acetylmorpholin-2-yl)methyl]-2,6-dimethoxypyrimidine-4-carboxamide
(3aR,7aS)-2-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
2-{2-[4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]ethyl}phenol
4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperazin-2-one
1-[(2-{[(4-ethyl-5-methylpyrimidin-2-yl)amino]methyl}phenyl)methyl]pyrrolidin-2-one
1-{4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepan-1-yl}-2-(2-phenyl-1H-imidazol-1-yl)ethan-1-one
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[(3-methylpyridin-4-yl)methyl]amine
ethyl 4-[(4-chlorophenyl)methyl]-1-[(4-fluorophenyl)carbamoyl]piperidine-4-carboxylate
2-[1-(cyclohexylmethyl)-4-(pyridin-4-ylmethyl)piperazin-2-yl]ethan-1-ol
4-{[3-(thiophene-2-carbonyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(thiophene-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
5-methyl-1-{2-oxo-2-[3-(pyrimidin-4-yl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
9-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(4-methoxyphenyl)ethyl]-1,5-dimethyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
{3-[5-(4,5-dimethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]propyl}(methyl)amine
N-(2,3-dichlorophenyl)-4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carboxamide
3-ethyl-N-[2-(5-methylfuran-2-yl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
N-(2-methoxyethyl)-4-methyl-3-{[methyl(propan-2-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-[4-chloro-3-({[(1-hydroxycyclohexyl)methyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
2-methyl-5-[2-(piperazin-1-ylmethyl)phenyl]quinoline
1-{4-[2-(furan-2-yl)azepane-1-carbonyl]phenyl}pyrrolidin-2-one
2,5-difluoro-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
3-(5-methylfuran-2-yl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}-1H-pyrazole-5-carboxamide
3-(aminomethyl)-N-[4-(4-methoxyphenyl)phenyl]pyrrolidine-1-carboxamide
(3S,9aR)-8-[(5-chlorothiophen-2-yl)methyl]-3-(1H-imidazol-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]-4-sulfamoylbenzamide
2-ethyl-N-methyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]pyrimidine-5-carboxamide
2-{2-[1-(2-phenoxyethyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[1-(3-methylpyridin-2-yl)propan-2-yl]amine
7-(2-methoxyphenyl)-2-[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-1-[2-methyl-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
1-ethyl-3-(naphthalen-1-ylmethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione