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1-({[5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}methyl)cyclohexan-1-ol
4-[3-(3,4-diethoxyphenyl)propyl]-4H-1,2,4-triazole
2-(2-hydroxyethyl)-9-(thiophen-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4S)-1-[(4-methoxypiperidin-1-yl)sulfonyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
1-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}-3-(2-methylphenyl)pyrrolidin-3-ol
(1R,5R)-6-(cyclopropylmethyl)-3-[3-(difluoromethoxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
5-{[4-(4-benzyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]methyl}-2-methylpyrimidine
1-(1-methyl-1H-pyrazole-3-carbonyl)-3,3-diphenylpiperidine
N-[(2R,3R)-2-methoxy-1'-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
4-ethyl-3-(1-{6-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(3aS,6aS)-2-cyclopentanecarbonyl-5-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-cyclopropyl-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
N-benzyl-N,1-dimethyl-5-[(prop-2-en-1-yl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-(3-methoxypropyl)-2-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
[(2S)-1-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)pyrrolidin-2-yl]methanol
N-(3-chloro-4-methoxyphenyl)-3-[1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-3-yl]propanamide
1-[(2-methyl-1,3-benzothiazol-6-yl)sulfonyl]azepan-4-amine
N-({1-[(3,4-dimethoxyphenyl)methyl]piperidin-3-yl}methyl)-4-fluorobenzamide
1-[2-(4-methoxybenzenesulfonamido)ethyl]-5-oxopyrrolidine-3-carboxylic acid
2-[2-(4-fluorophenyl)ethyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
2-[(3-propylmorpholin-4-yl)methyl]benzonitrile
N-butyl-3-{[(4,6-dimethylpyrimidin-2-yl)methyl]sulfamoyl}benzamide
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-[(3-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
9-(2-hydroxyethyl)-1-methyl-4-(5-methyl-1,3,4-thiadiazol-2-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(2,5-dimethylphenoxy)-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
4-chloro-N,N-dimethyl-5-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)-1,3-thiazol-2-amine
N-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-(oxan-4-yl)piperidine-3-carboxamide
1-{1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}-N,N-diethylpyrrolidin-3-amine
7-(1-benzothiophen-3-yl)-4-[2-(morpholin-4-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N,N-diethyl-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
(3aR,6aR)-2-cyclopropanecarbonyl-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-[5-(2-ethylpyrimidin-5-yl)-4-phenyl-1H-imidazol-1-yl]propanoic acid
2-(propan-2-yl)-9-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-5-(propan-2-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,2-oxazole-3-carboxamide
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrrolidine-3-carboxamide
5,7-dimethyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
6-methoxy-3-[(3-oxo-4-phenylpiperazin-1-yl)methyl]-1,2-dihydroquinolin-2-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-chloro-4-fluoro-1-benzothiophene-2-carboxamide
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(2-oxopyrrolidin-1-yl)butanamide
2-(1-ethylpiperidin-4-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
methyl 4-({5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazol-3-yl}formamido)butanoate
1-(carbamoylmethyl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)piperidine-4-carboxamide
1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidine-3-carboxamide
3-methyl-1-(2-methylpropyl)-4-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-2-(1H-pyrazol-1-yl)acetamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
6-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]-1H-indazole